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N-{[7-methoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-5-methylthiophene-2-carboxamide
1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-cyclopentyl-N-[cyclopropyl(3-methylpyridin-2-yl)methyl]pyrimidin-2-amine
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1,8-naphthyridine-2-carboxamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[3-(3-methylphenyl)phenyl]urea
4-[(1R,7S)-3-(2-ethoxyethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]piperazine-1-carboxamide
3-{[3-(2-methoxyethyl)-1-(4-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1-methyl-1H-indole
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}methyl)-5-methylpyridine-3-carboxamide
1-({4-[(2-fluoro-5-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2-methylbutyl)propanamide
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
6-(methoxymethyl)-2-[4-({methyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
2-benzyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,3-thiazole-4-carboxamide
1-(4-{4-azaspiro[2.5]octan-4-ylmethyl}-2-methoxyphenoxy)-3-(diethylamino)propan-2-ol
(2R,3R)-3-amino-1'-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(2-fluoro-5-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N,N-dimethyl-3-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]aniline
4-(3-fluoropropyl)-2-(6-methoxynaphthalen-2-yl)morpholine
2-{[(2-methyl-1,3-thiazol-4-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
2-(4-ethylpiperazin-1-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyridine-4-carboxylic acid
ethyl 4-(3-cyano-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)butanoate
(1R,5R)-3-methanesulfonyl-6-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperazin-1-yl}phenol
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(morpholin-4-yl)propan-1-one
1-(2-methoxyacetyl)-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-3-carboxamide
3-{1-[(3-chloro-5-fluorophenyl)methyl]piperidin-3-yl}propanoic acid
(3R)-1-(3-fluoropyridin-2-yl)-3,4,4-trimethylpyrrolidin-3-ol
4-(2,4-dioxoimidazolidin-1-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-ethyl-2-methyl-N-(pyridin-4-ylmethyl)-1-benzofuran-5-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]butan-1-one
N-(cyclopent-3-en-1-yl)-7-(furan-3-carbonyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1H-pyrazol-4-yl)propan-1-one
(2S,4R)-4-amino-1-[(2,5-dimethoxyphenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-({3-methyl-7-[3-(prop-2-en-1-yloxy)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
1-ethyl-4-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}piperazine-2,3-dione
4-methyl-2-[1-(oxane-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-ethyl-5-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}pyrimidin-2-amine
2-(3-methoxyphenyl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
ethyl 1-[(5-methylthiophen-2-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
2-{[1-(2-fluoro-6-methoxybenzoyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
1-cyclohexyl-4-(1-ethyl-1H-pyrazole-4-carbonyl)piperazine
2-({2-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-(hydroxymethyl)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-3-ol