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1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
(3S,5R,9R)-11-(2-chlorobenzoyl)-5-hydroxy-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
(1R,5R)-N,N-dimethyl-6-(4-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-3,5-dimethyl-1H-pyrazole
2-{1-[(4-fluorophenyl)methyl]-4-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
3-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
7-[(2,3-dimethoxyphenyl)methyl]-6-oxo-N-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
N,N-dimethyl-3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrazin-2-amine
1-{3-[bis(2-hydroxyethyl)amino]propyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
4-ethyl-1-[2-(naphthalen-2-yl)acetyl]-1,4-diazepan-5-one
2-fluoro-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-5-sulfamoylbenzamide
[(2R)-1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-2-yl]methanol
2-(4-{[1-(prop-2-yn-1-yl)-1H-indol-3-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-methyl-N-[2-(pyridin-2-yl)ethyl]benzamide
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-1-benzothiophene-2-carboxamide
2-amino-4-(furan-3-yl)-6-(2-methylpropyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-chloro-4-[(1-cyclobutylpiperidin-4-yl)oxy]-N-cyclopentylbenzamide
2-{[5-(2,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}-N-methylacetamide
1-(1H-imidazol-4-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
1-(2-cyclohexylethyl)-3-[(cyclopropylamino)methyl]-3-hydroxypiperidin-2-one
4-{[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
8-(4-propylpyrimidine-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-methyl-4-{[2-(2-methylphenyl)pyrrolidin-1-yl]methyl}-1-(prop-2-en-1-yl)-1H-pyrazole
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
8-[(5-cyclopentylthiophen-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}quinoline-2-carboxamide
(3S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N,N-dimethyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
4-(1H-imidazol-2-ylmethyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(3aR,6aR)-2-[6-(methoxymethyl)pyrimidin-4-yl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
(1S,9S)-11-(2-cyclopropyl-4-hydroxypyrimidine-5-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
5-methyl-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-benzoyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3S,9R)-11-(2,5-difluorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-N-ethylpyrrolidine-3-carboxamide
(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)methanamine
N-{[7-(1,3-benzothiazol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
5,5-dimethyl-3-[2-oxo-2-(2-phenylmorpholin-4-yl)ethyl]-1,3-oxazolidine-2,4-dione
2-(3,4-dichlorophenyl)-4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)morpholine
(2S,4R)-4-[3-chloro-4-(pyrrolidin-1-yl)benzamido]-N,1-dimethylpyrrolidine-2-carboxamide
5-benzyl-5-(1-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}piperidin-4-yl)imidazolidine-2,4-dione
4-[6-(3-methyl-3-phenylpiperidin-1-yl)pyrazine-2-carbonyl]morpholine
3-[2-(4-methoxyphenyl)ethyl]-3H,4H-pyrido[2,3-d]pyrimidin-4-one
ethyl N-{[(2S,4S)-4-fluoro-1-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]pyrrolidin-2-yl]methyl}carbamate
3-(pyridin-3-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}propan-1-one
2-hydroxy-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]pyridine-3-carboxamide
(1R,9S)-5-amino-3-[2-(methylsulfanyl)phenyl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
1-{6-[4-(methylsulfanyl)phenyl]pyridin-2-yl}piperazine
N-(1-cycloheptylpiperidin-3-yl)-3-(2-fluorophenyl)propanamide