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4-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanoic acid
4-benzyl-1-[(2-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S)-2-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)propanamide
6-methyl-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-{2-[4-hydroxy-3-(prop-2-en-1-yl)phenyl]-1H-imidazol-1-yl}-N-(propan-2-yl)acetamide
2-(2,3,4-trimethoxyphenyl)pyridine-3-carboxamide
N-(2-{5-[(2E)-pent-2-en-3-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)acetamide
2-[4-(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)quinazolin-2-yl]ethan-1-amine
1-(2-cyclopentylacetyl)-3-ethylpiperidine-3-carboxylic acid
4-{2-[1-butyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]propyl}morpholine
[4-({4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
3-(1H-pyrazol-1-ylmethyl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]benzamide
N-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
2-({3-[butyl(methyl)carbamoyl]phenyl}amino)acetic acid
1-tert-butyl-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
{4-benzyl-1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}methanol
N,1-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4R)-4-amino-1-{2-[(1,3-benzothiazol-2-yl)amino]acetyl}-N-methylpyrrolidine-2-carboxamide
4-(2-methyl-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}propan-2-yl)morpholine
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)methylamine
4-(2,2-diphenylethyl)-3-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]piperazin-2-one
3-{[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}-1-phenylpropan-1-ol
1-{1'-[2-(pyridin-3-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
methyl 4-(5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]methanesulfonamide
1-benzyl-2-[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]piperidine
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(3-methylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-methyl-7-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-[2-(1-{2-[4-(dimethylamino)phenyl]acetyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
1-[(3S,4R)-1-(1-benzothiophene-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-{[5-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methyl-1,3,4-oxadiazole
(3S)-4-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3-ethylmorpholine
2,6-dimethyl-4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]quinoline
2-(2,5-dioxoimidazolidin-1-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
5-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-2-(2-methylphenyl)pyrimidine
1-methyl-4-[2-(pyrrolidin-1-yl)benzoyl]-1,4-diazepan-6-ol
2-hydroxy-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-propyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrimidin-4-amine
(4aS,8aR)-6-[2-(5-amino-1,3,4-thiadiazol-2-yl)acetyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
2-(furan-2-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxoacetamide
2-benzyl-8-(1,3-dihydroxypropan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(1-hydroxycyclohexyl)methyl]propanamide
4,6-dimethyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
1,3-dimethyl-6-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[2-(1-methylpyrrolidin-3-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-4-carbonitrile