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1,3-dimethyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}ethan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(oxolan-2-ylmethyl)benzamide
2-[4-(4-{[2-(1H-imidazol-1-yl)ethyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-yl]phenol
3-benzoyl-1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methyl-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
8-chloro-N-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carboxamide
(4S)-3,3,4-trimethyl-1-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]piperidin-4-ol
1-[4-(ethylsulfanyl)phenyl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(2S)-N2-[1-(2,5-difluorophenyl)cyclopropyl]pyrrolidine-1,2-dicarboxamide
2-(2,1-benzoxazole-3-carbonyl)-8-methyl-2,8-diazaspiro[4.5]decane
4-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-2-yl}pyridine
1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4-diazepane-6-carboxylic acid
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
4-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-5-methyl-2-(2-methylphenyl)-1,3-oxazole
2-(2-methyl-1H-1,3-benzodiazol-1-yl)pyridin-3-ol
N-cyclopentyl-1-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-({ethyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
N-methyl-N-(oxan-2-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
3-hydroxy-1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
6-(2-aminoethyl)-N-[2-(4-methoxyphenyl)ethyl]pyrimidin-4-amine
[(1-cyclohexylpiperidin-3-yl)methyl]({[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
N-[(4-hydroxyazepan-4-yl)methyl]-2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
(3R,4R)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
3-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-N-(pyridin-3-yl)benzamide
3-[5-({3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}methyl)thiophen-3-yl]prop-2-yn-1-ol
9-(3-ethyl-1,2-oxazole-5-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-oxopentanamide
N-[4-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-3-phenylpropanamide
4-[(4-fluorophenyl)methyl]-1-(5-methylpyrazine-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5,6-dimethyl-2-oxo-N-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-methylacetamide
2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}-N-(propan-2-yl)acetamide
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(3-hydroxy-3-methylbutyl)benzamide
(2S)-2-{[5-(2,6-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}propanamide
1-methyl-4-{5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-phenyl-1H-1,2,4-triazol-1-yl}piperidine
2-(3-chloro-4-fluorophenoxy)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
N-[3-(morpholin-4-yl)propyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-methoxy-N-{[5-(3-phenylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
2-methyl-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}-2,3-dihydropyridazin-3-one
3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)piperidin-3-ol
1-[4-(1-hydroxypropyl)piperidin-1-yl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-amino-4-(3,5-dimethyl-1H-pyrazol-4-yl)-5-methyl-6-phenylpyridine-3-carbonitrile
6,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline