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3-[(2,4-difluorophenyl)methyl]-1-(3,6-dimethylpyrazin-2-yl)piperidine-3-carboxylic acid
1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-5-[2-(1H-imidazol-4-yl)-1-(1H-pyrrol-1-yl)ethyl]-1H-1,2,4-triazole
3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propanamide
2-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-1-phenylethan-1-ol
5-{1-[2-(ethylsulfanyl)ethyl]-1H-1,2,3-triazol-4-yl}-2-methoxybenzoic acid
4,6-dimethyl-2-{4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazin-1-yl}pyrimidine
3-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]propan-1-one
3,3-dimethyl-1-({5-[(2,3,6-trifluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)naphthalene-1-carboxamide
6-(2-butoxy-4-fluorophenyl)pyrazine-2-carboxylic acid
(1S,5R)-6-benzyl-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-2,1,3-benzoxadiazole
8-(2,6-dimethoxypyridine-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N,5-dimethyl-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
N-(oxolan-2-ylmethyl)-4-({[2-(1,3-thiazol-2-yl)ethyl]carbamoyl}amino)benzamide
1-[4-(furan-2-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-3-(pyrrolidin-1-yl)propan-1-one
1-(1-benzothiophene-2-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
5-{[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}quinoxaline
methyl({[1-(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl})amine
(1R,7S)-3-(2,2-dimethylpropyl)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[4-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}amino)-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)-2-methylpropan-1-ol
5-(2-ethoxypyridin-3-yl)-2,3-difluorophenol
5-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}quinoxaline
N-ethyl-4-methyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]-1,3-thiazol-2-amine
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
5-(2,4-difluorophenoxymethyl)-N-[2-(methylamino)ethyl]-1,2-oxazole-3-carboxamide
1,3,7-trimethyl-N-(2,2,2-trifluoroethyl)-1H-indole-2-carboxamide
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
6-oxo-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1-(2-phenylethyl)piperidine-3-carboxamide
9-[(2-ethylphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-1-[4,5-dimethyl-2-(1H-1,2,3,4-tetrazol-1-yl)thiophene-3-carbonyl]-N-methylpyrrolidine-2-carboxamide
9-[2-(1H-imidazol-2-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
4-chloro-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-3-carboxamide
[(8-methoxyquinolin-5-yl)methyl](methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
4-[1-methyl-3-(4-methylthiophen-3-yl)-1H-1,2,4-triazol-5-yl]morpholine
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(propan-2-yl)amino]methyl}piperidin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
1-cyclopentyl-5-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
6-(2-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-oxoethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-[4-(2-methylpyridin-4-yl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
5-{2-[bis(propan-2-yl)carbamoyl]-3-methoxyphenyl}-N-methylfuran-2-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrrole-2-carboxamide
1-{2-[5-(morpholine-4-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
5-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-[(propan-2-yl)sulfamoyl]-5-(propylamino)benzamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
2-ethyl-4-methyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1,3-oxazole-5-carboxamide