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1-{[2-(cyclopentyloxy)phenyl]methyl}pyrrolidin-3-amine
7-[2-hydroxy-6-(trifluoromethyl)pyridine-3-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
methyl 3-(4,5,6,7-tetrahydro-2H-indazol-3-ylformamido)propanoate
5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
5-[3-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
N-({1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
N2-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-cyclopropyl-4-{6-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}pyrrolidin-2-one
6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazolo[1,5-a]pyrimidine-2-carboxylic acid
4-{2-[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3-thiazol-2-amine
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-1,2-dihydroquinazoline-4-carboxamide
1-ethyl-3-(propan-2-yl)-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
8-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(4-chlorophenyl)-1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-ol
N-{[7-(1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-methoxy-2-phenylacetamide
N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amine
6-[2-(4-hydroxyphenyl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{4-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
ethyl 1-(ethanesulfonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-(trifluoromethyl)morpholine
5-[5-(2-chlorophenyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
8-(butan-2-yl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
N-[(5-fluoro-2-methylphenyl)methyl]-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
4-chloro-1-ethyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-pyrazole-5-carboxamide
3-(azepane-1-carbonyl)-1-methyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-4,5,6,7-tetrahydro-1H-indazole
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(methylamino)ethan-1-one
ethyl 2-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,3-thiazole-4-carboxylate
N,N-diethyl-1-[6-(2-methoxyphenyl)pyridazin-3-yl]pyrrolidin-3-amine
(2S)-2-amino-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(1,3-thiazol-4-yl)propanamide
(3R,4R)-1-[(2,4-difluorophenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-methyl-2-(methylamino)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-4-carboxamide
2-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)-N-(pyrazin-2-yl)acetamide
3-(2-{1-[2-(dimethylamino)benzoyl]piperidin-2-yl}ethyl)phenol
(1S,5R)-3-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
3-(1H-pyrazol-1-ylmethyl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]benzamide
2-[(4-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}piperidin-1-yl)methyl]pyridine
4-[4-(5-chloro-2-methylpyrimidine-4-carbonyl)piperazin-1-yl]quinazoline
7-cyclopentyl-2-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-6-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyridine-3-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(naphthalen-1-yl)ethyl]propanamide
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
1-(4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
4-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-5-ethyl-6-methylpyrimidin-2-amine
9-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
3-methoxy-2-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol