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6-phenyl-3-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
3-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]pyridin-1-ium-1-olate
1-{1-[2-(2-hydroxyphenyl)acetyl]piperidin-3-yl}pyrrolidin-2-one
3-{1-[2-amino-6-(dimethylamino)pyrimidin-4-yl]piperidin-4-yl}-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,7-dimethylimidazo[1,2-a]pyridine-3-carboxamide
3-[({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)methyl]pyrrolidin-3-ol
4-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}-2-(propan-2-yl)pyrimidine
(2R)-N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-5-oxopyrrolidine-2-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-2-methylpyridine
methyl 2-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetate
N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(4-propanoylphenoxy)acetamide
N-methyl-3-(2-oxopiperidin-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
3-methyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(6-phenoxypyridin-3-yl)urea
methyl 3-[(3S,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
2-(4-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)ethan-1-ol
N-[(3S,4R)-1-(4-aminopyrimidin-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-ethyl-N-[(5-methylfuran-2-yl)methyl]-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
(1R,5R)-6-benzyl-3-(3,4-difluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanoyl]piperidine-3-carboxamide
N-benzyl-1-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]-N-methylpiperidin-3-amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,3-dimethylbutanamide
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[3-fluoro-5-(trifluoromethyl)phenyl]-3-(propan-2-yl)urea
3-(4-methylphenoxymethyl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-pyrazol-1-yl)propan-1-one
(2E)-N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-(furan-2-yl)-N-[2-(piperidin-1-yl)ethyl]prop-2-enamide
2-(4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyrazine
1-cyclohexyl-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-2-(pyridin-4-yl)ethan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}acetamide
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
4-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}-N-methylbenzene-1-sulfonamide
N-benzyl-2-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
2-[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carbonyl]benzonitrile
2-{5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
2-(2,6-dimethoxyphenyl)-2-{methyl[2-(pyrrolidin-1-yl)ethyl]amino}acetic acid
5-(2,3-dihydro-1-benzofuran-7-carbonyl)-3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]-1H-imidazole
(3S,4S)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}pyrrolidin-3-ol
1-{4-[(3-chlorophenyl)methyl]-5-oxo-1,4-diazepan-1-yl}-4-(4-fluorophenyl)butane-1,4-dione
(3R,4R)-4-amino-1-({2-[(benzenesulfonyl)methyl]phenyl}methyl)piperidin-3-ol
2-amino-4-[4-(dimethylamino)phenyl]-6-propyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl](propan-2-yl)amine
2-{4-[3-(4-chlorobenzoyl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
2-{4-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]morpholin-3-yl}-1-(4-methylpiperazin-1-yl)ethan-1-one
(2S,4S)-N,N-diethyl-4-(2-hydroxyacetamido)-1-[2-(2-methylphenyl)acetyl]pyrrolidine-2-carboxamide
1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-(thian-4-yl)piperazine
3-{2-[3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-2,6,6-trimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indol-4-one