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1-[1-(cyclohex-1-en-1-yl)ethyl]-3-(1,3-dihydro-2-benzofuran-5-yl)urea
(1R,5R)-3-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-[methyl(pyrazin-2-ylmethyl)amino]-2-[3-(2-methylpropoxy)phenyl]acetic acid
8-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
2-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methylpyrimidin-2-amine
5-ethyl-N-[(1-ethylpyrrolidin-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(3-chlorophenyl)-4-(1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidin-3-yl)piperazine
3-{2-[5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1H-1,2,3-benzotriazol-5-yl)-5-oxopyrrolidine-3-carboxylic acid
N-[2-(2,4-dimethylphenoxy)ethyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
[(3R,4R)-1-(2-chloro-4-fluorobenzoyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
(2R)-2-{2-[6-(dimethylamino)pyridin-3-yl]-1H-imidazol-1-yl}-3-phenylpropan-1-ol
2,3-dimethyl-7-{[4-(thian-4-yl)piperazin-1-yl]methyl}-1H-indole
3-(3-cyanopiperidine-1-carbonyl)-N-[2-(1H-imidazol-1-yl)ethyl]benzene-1-sulfonamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-[3-(trifluoromethyl)benzenesulfonyl]piperidine
N-[(1-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
N-(1-benzothiophen-5-ylmethyl)-3-(2,5-dioxoimidazolidin-4-yl)propanamide
2-{1-benzyl-5-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
(2E)-N-({7-[1-(4-hydroxy-3-methoxyphenyl)propan-2-yl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
4-[3-(3,4-dimethoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]thiomorpholine
N-[(2S,4R,6S)-2-ethyl-6-[2-(2-phenylethynyl)phenyl]oxan-4-yl]acetamide
9-(pyrimidin-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-cyano-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}benzamide
2-methoxy-2-methyl-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
5-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]quinoline
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-(2-methoxy-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3-(4-ethoxyphenoxymethyl)-1-ethyl-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
2-(4-methylpyrimidine-5-carbonyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-2,3-dimethyl-N-[(3S)-2-oxoazepan-3-yl]-1H-indole-5-carboxamide
5-(2-cyclopentyl-2-phenylacetyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[benzyl(methyl)amino]-N-(pyridin-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
N-(3-cyanophenyl)-4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazine-1-carboxamide
(2S,4S)-1-methyl-4-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]pyrrolidine-2-carboxylic acid
4-(4-ethyl-1H-pyrazol-5-yl)-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperidine
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
1-cyclopentyl-4-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazine
3-(1H-imidazol-1-yl)-1-[3-(4-methylphenoxymethyl)piperidin-1-yl]propan-1-one
N-(1H-indol-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-(2-amino-6-methylpyrimidin-4-yl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylic acid
4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-8-thia-4,6-diazatricyclo[7.6.0.02,7]pentadeca-1(9),2(7),5-trien-3-one
1-(2-methoxypyridin-3-yl)-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]pyridine-2,4-diol
(2R,3R,6R)-5-(2,3-difluorobenzoyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
1-[4-(difluoromethoxy)benzoyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
5-(3-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-3-oxopropyl)-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one