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8-methoxy-N-methyl-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(4-hydroxyphenyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
(2S,4R)-4-amino-N,N-diethyl-1-[4-methyl-3-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxamide
1-(4-{2-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
2-(3-phenylpropyl)-5-(pyrrolidine-1-carbonyl)-1,3-benzoxazole
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl]-2-methoxyacetamide
{[(1R,5S,6S)-3-[2-chloro-5-(piperidin-1-yl)benzoyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
ethyl 5-(1H-imidazol-2-ylmethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(cyclopropylmethyl)-8-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(1H-1,3-benzodiazol-2-yl)-1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
N-[2-(dimethylamino)ethyl]-6-methyl-2-oxo-4-[2-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-4,5,6,7-tetrahydro-1H-indazole
1-cyclopentanecarbonyl-3-(2-phenylethyl)piperidine
4-phenyl-1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)piperidin-4-ol
8-methyl-N-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyridine-2-carboxamide
4-[hydroxy(pyridin-2-yl)methyl]-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
1-{3-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}ethan-1-one
9-[(5-ethylpyridin-2-yl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(1H-pyrazole-3-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[2-(3-fluorophenyl)piperidin-1-yl]ethan-1-one
2-(3-methyl-1H-1,2,4-triazol-5-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-phenyl-1H-pyrazole-4-carboxamide
N-benzyl-N-methyl-3-{[(thian-4-yl)amino]methyl}pyridin-2-amine
(2S,4S)-N-ethyl-1-(oxan-4-yl)-4-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamido]pyrrolidine-2-carboxamide
1-[(3R,4S)-3-(dimethylamino)-4-phenylpyrrolidin-1-yl]-3-methanesulfonylpropan-1-one
4-(1-methyl-1H-imidazol-2-yl)-1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]piperidine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-{1-[(2-fluorophenyl)methyl]-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-N-(pyridin-2-yl)benzamide
2-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[6-(2-aminoethyl)pyrimidin-4-yl]-N-benzyl-N-methylpiperidin-4-amine
3-{[1-(6-methylpyridine-2-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-(3-methylpyridin-4-yl)-1,4-diazepane
2-[1-(2-ethoxypyridine-3-carbonyl)piperidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4-sulfamoylbutanamide
(2S,4S)-4-amino-1-(3-hydroxy-2-methylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[1-(oxan-4-yl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
4-[(3-methoxyphenyl)methyl]-1-[(3-methylphenyl)methyl]-1,4-diazepan-5-one
5-fluoro-3,8-dimethyl-2-[4-(pyrimidin-5-ylmethyl)piperazin-1-yl]quinoline
4,6-dimethyl-2-oxo-N-[3-(2-phenylacetamido)phenyl]-2H-pyran-5-carboxamide
5-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,3-oxazole-4-carboxamide
N-(2-ethoxyphenyl)-3-oxo-3-[2-(2-phenylethyl)pyrrolidin-1-yl]propanamide
1-[(3,4-difluorophenyl)methyl]-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-[2-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-1-yl]acetic acid
8-[(2R)-2,3-dihydroxypropyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one