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N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2,7-dioxo-1,3-diazepane-4-carboxamide
(2R,3R)-3-[4-(2-fluorophenyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-(pyridin-2-yl)pyrimidin-2-amine
2-{8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]phenol
{3-[2-(4-chloro-2-fluorophenyl)-1H-imidazol-1-yl]phenyl}methanol
N-[(2-fluorophenyl)methyl]-2-{[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]amino}acetamide
4-(4-tert-butylbenzenesulfonyl)piperazine-2-carboxylic acid
1-[(2R,3R)-3-(dimethylamino)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-hydroxy-3-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)-1-(2-phenylethyl)piperidin-2-one
N-(4-fluoro-2-methylphenyl)-3-[1-(3-methylbut-2-enoyl)piperidin-3-yl]propanamide
3-({5-acetyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}formamido)-N-(2,5-dimethylphenyl)propanamide
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-3-carboxamide
(2E)-N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(4-methoxyphenyl)prop-2-enamide
1-[(2S)-2-phenylbutanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}cyclopentanamine
1-[(2S)-oxolan-2-ylmethyl]-4-phenyl-5-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
6-(cyclopentylmethyl)-2-(3-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-(oxolan-3-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
1-{2-[(5-methylhex-5-en-2-yl)amino]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
(1R,7S)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(4-fluorophenyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-(oxolan-2-ylmethyl)urea
2-(3-chlorophenoxy)-1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)propan-1-one
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-{[(thian-4-yl)amino]methyl}pyridin-2-amine
(1R,5R)-6-(cyclobutylmethyl)-3-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(furan-2-yl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H-pyrazole-4-carboxamide
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
methyl 6-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-3-(1,3-dimethyl-1H-pyrazole-5-amido)thieno[2,3-b]pyridine-2-carboxylate
7-(2,2-dimethylpropyl)-2-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-6-[4-oxo-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
(3S,9R)-11-(3-methylbenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
4-({2-[1-(3-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-cyclohexyl-7-[(3-hydroxybutyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
3-(3,4-difluorophenyl)-1-{3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]morpholin-4-yl}propan-1-one
N-[(3-fluoro-4-methoxyphenyl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
5-[1-(furan-2-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(4-methoxyphenyl)-1-benzofuran-2-carboxamide
5-amino-N-[3-(1,3-benzothiazol-2-yl)propyl]-1H-pyrazole-3-carboxamide
6-(2-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}ethyl)-2-methylpyrimidin-4-ol
1-({4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)piperidine
2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
2-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]pyrrolidin-2-yl}pyridine
3-(3-chloropyridin-2-yl)-3,9-diazaspiro[5.6]dodecan-10-one
5-{4-[(3-chloro-4-methoxyphenyl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-[(6-ethylpyrimidin-4-yl)amino]-1-(2-methoxyethyl)pyrrolidin-2-one
N-cyclopropyl-4-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperazine-2-carboxamide
N-(oxan-3-ylmethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(azepan-1-yl)ethyl]-5-ethyl-2-methylpyrimidin-4-amine
methyl[(1-phenylpyrrolidin-3-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine