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4-benzyl-1-methyl-3-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(2E)-2-methylbut-2-en-1-yl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
9-(3-cyclopentylpropanoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
3-(furan-2-yl)-N-[(3-methyloxetan-3-yl)methyl]benzamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propane-2-sulfonamide
7-(5-chloropyridin-2-yl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-(2,4-difluorophenoxy)-N-methylacetamide
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(1-methyl-1H-pyrazol-3-yl)-2-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
2-(adamantan-1-yl)-N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}acetamide
5-ethyl-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-1,3-oxazole-4-carboxamide
5-chloro-2-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
N-(2-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
[(5-chloro-2-fluorophenyl)methyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
7-(5-methylthiophen-2-yl)-4-(pyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
2-(2-aminoethyl)-N-[(1R,2S)-2-phenylcyclopropyl]quinazolin-4-amine
3-(2H-1,3-benzodioxol-5-yl)-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-(2,5-dioxoimidazolidin-4-yl)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylpropanamide
5-(3-fluorophenyl)-N-methyl-N-(oxan-2-ylmethyl)-1,2,4-triazin-3-amine
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-(propan-2-yl)propanamide
1-[2-(1H-imidazol-4-yl)ethyl]-4-(2-methyl-1-benzothiophen-3-yl)-1H-1,2,3-triazole
N-[3-(propan-2-yloxy)propyl]-3,4-dihydro-2H-1-benzopyran-3-amine
(1R,5S)-3-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-3,8-diazabicyclo[3.2.1]octane
(4aR,7aS)-1-{2-[(2-methylpyridin-3-yl)oxy]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[2-(morpholin-4-yl)ethyl]piperidine-3-carboxamide
3-cyclohexyl-N-(cyclopropylmethyl)-N-(2-methoxyethyl)-1H-pyrazole-4-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(1H-indol-3-yl)propanamide
4-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperazin-1-yl]-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
(1R,2R)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-phenylcyclopropane-1-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]pyrimidin-4-amine
2-(4-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
5-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
5-(2-methoxy-4-methylphenoxymethyl)-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide
1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
2-(dimethylamino)-7-(1-ethyl-1H-pyrazole-3-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
methyl 3-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}benzoate
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(naphthalen-1-ylmethyl)piperidine
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)furan-3-carboxamide
dimethyl({[(1R,5S,6R)-3-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
3-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-phenyl-N-(1-{1-[3-(1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
2-methyl-N-{3-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]phenyl}propanamide
2,7,8-trimethyl-4-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]quinoline
(3aS,6aS)-2-(6-ethyl-2-methylquinoline-4-carbonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(1H-indol-3-yl)acetamide