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(1S,5R)-3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(pyridin-3-yl)-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
2-(3-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)acetamide
(9-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}-3,9-diazaspiro[5.5]undecan-1-yl)methanol
5-[3-(3-methylphenoxy)azetidine-1-carbonyl]isoquinoline
N-(4-cyclohexylphenyl)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
5-chloro-2-(2-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
4-(5-{3-fluoro-7-methylimidazo[1,2-a]pyridin-2-yl}-3-methyl-1H-1,2,4-triazol-1-yl)-1-methylpiperidine
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]propanoic acid
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2,3-dihydro-1H-inden-2-yl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
(3S,9aR)-8-(cyclopropylmethyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({7-[2-(1H-indol-3-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
5-cyclopropyl-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1,3,4-oxadiazol-2-amine
methyl 3-{[(3-methylthiophen-2-yl)formamido]methyl}-5-(quinoline-8-sulfonamido)benzoate
methyl 4-[2-amino-3-cyano-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]thiophene-2-carboxylate
N-methyl-4-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-[4-(2-methoxyphenyl)benzoyl]azepan-4-amine
2-(4-methylphenoxy)-1-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
4-{2-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylbenzene-1-sulfonamide
ethyl 1-{1-[(2-chlorophenyl)methyl]-7-oxoazepan-4-yl}piperidine-4-carboxylate
(3aS,6aS)-2-cyclopentyl-5-(dimethylsulfamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methoxy-5-{[(2-methylphenyl)methyl](oxolan-2-ylmethyl)carbamoyl}benzoic acid
methyl({4-[2-(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-2-yl)ethoxy]phenyl}methyl)(thiophen-2-ylmethyl)amine
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methanesulfonylpiperidine
ethyl 4-[3-({[2-(2-fluorophenyl)ethyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
3-chloro-N-(1,4-dioxan-2-ylmethyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
(1S,5R)-3-[(3-chlorophenyl)methanesulfonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(trifluoromethyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}morpholine
2-(methylsulfanyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-3-carboxamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-({ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-N-(1-methyl-1H-1,2,4-triazol-3-yl)benzamide
dimethyl[1-(5-methylfuran-2-yl)-2-{4-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}ethyl]amine
8-[(3,5-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-[4-(dimethylamino)phenyl]propan-1-one
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[(2-fluorophenyl)methyl]acetamide
4-(5-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-(1-butyl-1H-imidazol-2-yl)-1-(5-chloro-2-methylbenzoyl)piperidine
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(4-methyl-3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1,3,5-trimethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-4-carboxamide
(2S,4S)-4-(2,5-dimethylfuran-3-amido)-N,N-diethyl-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
2-{[4-(2,2-dimethoxyethyl)piperazin-1-yl]methyl}-4-methylphenol
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
8-(2,2-dimethylcyclopropanecarbonyl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{[(2-hydroxyethyl)(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)amino]methyl}-2,6-dimethylphenyl acetate
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol