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4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
1-{3-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}pyrrolidin-2-one
2-[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine-3-carbonyl]pyridine
N-butyl-4-{[2-(dimethylamino)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
9-[2-(morpholin-4-yl)acetyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aR,8aR)-2-(3-fluoropyridin-2-yl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
3-[(2-fluorophenyl)formamido]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
2-(1,4-dithiepan-6-yl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(dimethyl-1,2-oxazol-4-yl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4-(2-oxopyrrolidin-1-yl)benzamide
8-[(2S)-2-hydroxypropanoyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-methoxy-4-(morpholin-4-ylmethyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-(pyridin-2-ylmethyl)-4-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
4-[(2R,3R)-2-hydroxy-1'-(thiophene-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-2-one
4-{1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]azetidin-3-yl}morpholine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)propanamide
5,5-dimethyl-3-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3-oxazolidine-2,4-dione
N-[3-(4-methylbenzenesulfonamido)propyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
1-{2-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-5-(5-methyl-1,3-oxazole-4-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
6-(6-fluoroquinolin-8-yl)-N,N-dimethylpyridazin-3-amine
6-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2E)-3-(3-fluorophenyl)-1-[4-(3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
1-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]piperidine-3-carbonitrile
7-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
ethyl 4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]piperazine-1-carboxylate
N-methyl-N-(2-phenylethyl)-1-(quinolin-8-ylmethyl)piperidin-3-amine
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-[3-(2,5-dioxoimidazolidin-4-yl)propanoyl]-4-phenylpiperidine-4-carbonitrile
5-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-{4-[(3,5-dimethyl-1H-indol-2-yl)methyl]piperazin-1-yl}-5-methylpyrimidin-4-amine
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
(2E)-N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
methyl 1-[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]piperidine-4-carboxylate
N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
7-(cyclopropylmethyl)-2-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-methyl-2-(propan-2-yl)-N-[3-(pyridin-3-yloxy)propyl]-1,3-thiazole-5-carboxamide
N-[1-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
4-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-3-benzylpiperazin-2-one
2-(4-hydroxypiperidin-1-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
1-(furan-3-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
2-ethyl-7-methoxy-4-[(2-methyl-1H-imidazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[4-(trifluoromethyl)phenyl]methyl}amine
N-{[4-(furan-2-yl)phenyl]methyl}-N-methyloxan-4-amine
3-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]urea
1-(2-ethoxyethyl)-2-oxo-N-(propan-2-yl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-(2-methoxyphenoxy)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine