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(1R,5S,6R)-N-(2-hydroxyethyl)-3-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
5-(3-methoxyphenoxymethyl)-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-pyrazole-3-carboxamide
(3S,9aR)-3-benzyl-8-(4-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{2-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]ethyl}methanesulfonamide
N-benzyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-ethylpiperidine-3-carboxamide
1-(2-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-3,3-dimethylurea
1-methyl-2-(morpholin-4-yl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
methyl 4-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutanoate
2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]-1,4-dihydroquinolin-4-one
3-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-5-methyl-1H-indole-2-carboxylic acid
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-(propan-2-yloxy)ethan-1-one
3-[(dimethylamino)methyl]-1-(quinolin-2-yl)pyrrolidin-3-ol
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N,N-dimethylpiperidine-1-sulfonamide
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
1-{3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-1,2,5-thiadiazole-3-carboxamide
3-{2-[1-butyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
5-(1,3-benzothiazol-2-ylmethyl)-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-oxo-4-phenylbutanamide
[1-({1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
N-[2-(5-methylfuran-2-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine-3-carbonitrile
(2S,4R)-4-(furan-3-amido)-1-(3-methylbut-2-en-1-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(2-phenylpropyl)-8-(1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}ethan-1-one
(2,6-dimethylhept-5-en-1-yl)(ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
4-methoxy-N-{2-[7-(2-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-propoxyethan-1-one
methyl (3S)-2-(2-ethylpyrimidine-5-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-3-carboxylate
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-2-methylpyridine-3-carboxamide
N-(2-methoxyethyl)-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
(2S)-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-hydroxy-2-(methylamino)propanamide
3-[(dimethylamino)methyl]-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2,2-diphenylbutanenitrile
N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-methyl-N-{4-[(2-phenylethyl)carbamoyl]phenyl}-1,4-oxazepane-4-carboxamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3,4-dimethylphenyl)-1H-imidazole
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]urea
4-benzyl-3-ethyl-1-(3-hydroxypropyl)-1,4-diazepan-5-one
1-[4-(2,3-dihydro-1H-inden-2-yl)-6-hydroxy-1,4-diazepan-1-yl]-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
1-(2-chlorophenyl)-4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aR,7aS)-1-benzyl-4-[(4-hydroxy-3-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,8aR)-6-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-(4-fluorophenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2,2-dimethylcyclopropane-1-carboxamide
(2R,6R)-4-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]-1-[(2S)-2-hydroxy-2-phenylethyl]urea
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N-[2-({[1-(carbamoylmethyl)-2-methyl-1H-indol-3-yl]methyl}amino)ethyl]-4-fluorobenzamide