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1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-{5-amino-[1,2,4]triazolo[4,3-c]pyrimidin-7-yl}-4-(3-tert-butyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2,2-dimethylpropyl N-{[(3S,4S)-3-hydroxy-1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}carbamate
4-methyl-6-[3-(2-methylphenyl)piperidine-1-carbonyl]-1H,2H,3H-pyrazolo[3,4-b]pyridin-3-one
1-{2-[3-(3-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}imidazolidin-2-one
3-[4-(piperidine-1-carbonyl)phenyl]pyridin-4-amine
N-methyl-N-[2-(phenylsulfanyl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazin-1-yl}-4-phenylpyrimidine
(3-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-(1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
2-{1-[(3-methoxyphenyl)methyl]-4-(3-methoxypyrazin-2-yl)piperazin-2-yl}ethan-1-ol
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
(2S,4R)-4-amino-N-methyl-1-{3-methyl-1-phenyl-1H-thieno[2,3-c]pyrazole-5-carbonyl}pyrrolidine-2-carboxamide
5-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
N-(1-{7-[5-(methoxymethyl)furan-2-carbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
4-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
8-(1-methylpiperidine-2-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-[(3S,4S)-3-carboxy-4-cyclopropylpyrrolidin-1-yl]-5-chloropyridine-3-carboxylic acid
1-(5-chloropyridin-2-yl)-4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine
4-(2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-1-hydroxyethyl)phenol
3-(4-acetamido-3-methoxyphenyl)benzoic acid
2-butyl-4-methyl-N-(naphthalen-1-yl)-3-oxopiperazine-1-carboxamide
6-cyclopentyl-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]azetidin-3-yl}morpholine
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
5-ethyl-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)thiophene-2-carboxylic acid
N-methyl-3-[methyl({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amino]butanamide
N-[(5-chloro-1-benzothiophen-3-yl)methyl]-6-[(dimethylamino)methyl]pyrimidin-4-amine
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1,2,3-thiadiazole-4-carboxamide
2-methyl-4-{3-methyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,4-triazol-1-yl}pyridine
3-{4-[5-(2-methoxy-2-phenylacetamido)-1H-pyrazol-1-yl]piperidin-1-yl}propanamide
methyl 4-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}benzoate
1-[(2-chlorophenyl)methyl]-4-[(quinolin-8-ylmethyl)amino]pyrrolidin-2-one
N,N-dimethyl-4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-sulfonamide
5-[4-(1H-imidazol-1-yl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2,4-dimethylphenyl)-4-{furo[3,2-c]pyridin-4-yl}morpholine-2-carboxamide
5-methyl-5-phenyl-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-one
N-[(4-hydroxyazepan-4-yl)methyl]-2-methyl-4-phenylpyridine-3-carboxamide
7-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
6-{[(4aS,7aR)-4-benzyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,4S)-4-propyl-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}pyrrolidin-3-amine
1-{[3-(2,5-dimethoxyphenoxy)-2-fluorophenyl]methyl}pyrrolidine
1-(2,3-dihydro-1H-inden-2-yl)-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-[3-(5-methylfuran-2-yl)-1H-pyrazol-1-yl]acetamide
4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
(3R,4S)-1-(4-chloro-2-methoxybenzoyl)-4-(3-methoxyphenyl)pyrrolidin-3-amine