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({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
8-(2,2-dimethylpropyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-4-cyclopropyl-1-[3-(pyridin-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-ethyl-N,N-dimethyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,2,4-triazol-5-amine
3-cyclohexyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-(3-fluorophenoxymethyl)-N-[2-(morpholin-4-yl)ethyl]piperidine-3-carboxamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
8-(dimethyl-1,3-oxazole-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-[3-(methylsulfanyl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
{2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}urea
2,6-difluoro-3-methoxy-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
1-(5-{3-[(3,4-dimethoxyphenyl)amino]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
(3R)-3,4,4-trimethyl-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-ol
(4aS,7aR)-1-[(8-methoxy-2H-chromen-3-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyclopropanecarbonyl-1'-(1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
7-(cyclohexylmethyl)-2-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
4-[(2S)-2,3-dihydroxypropyl]-1-(2-phenylphenyl)piperazin-2-one
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[2-(2-oxopyrrolidin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyridine-2-carbonitrile
(5-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}furan-2-yl)methanol
(2R)-2-amino-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-phenylethan-1-one
ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
2-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
3-[2-fluoro-5-(trifluoromethyl)phenyl]-1-[(1S,2S)-2-hydroxycyclohexyl]urea
6-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-3-yl}-2-methylpyrimidin-4-ol
1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-propoxyethan-1-one
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-methyl-5-propylpyrimidine
(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N3-(butan-2-yl)-1-cyclopentyl-N5-[3-(methylsulfanyl)propyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-(3-methylbutyl)-8-[4-(2-oxopyrrolidin-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-5-(3-{[(quinolin-2-yl)amino]methyl}pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
(3aS,6aS)-5-[(3-chloro-4-fluorophenyl)methyl]-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-methyl-1H-pyrazol-1-yl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-methylbut-2-en-1-yl)piperidin-3-ol
(1R,5R)-6-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{[1-(furan-2-ylmethyl)piperidin-4-yl]formamido}-N,N-dimethyl-2-phenylacetamide
8-[(2S,3S)-2-amino-3-methylpentanoyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}-N-cyclopropyl-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
N-[6-(dimethylamino)-1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-2,3-dihydro-1H-isoindole-2-carboxamide
4-{[1-(furan-2-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]pyrrolidine-2-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
9-[3-(5-methylfuran-2-yl)butyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-ethoxy-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
3-(2-{4-phenyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-imidazol-5-yl}-1H-pyrrol-1-yl)pyridine