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2,2-dimethyl-N-{[1-(quinolin-4-ylmethyl)piperidin-3-yl]methyl}propanamide
7-[(2,3-difluorophenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1,3-dimethyl-4-{6-methyl-2-[2-(methylamino)pyrimidin-5-yl]quinoline-4-carbonyl}piperazin-2-one
4-[(3-methylphenyl)sulfanyl]-1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}piperidine
3-[2-(azepan-1-yl)-2-oxoacetamido]-N-(2-fluorophenyl)propanamide
2-(1-methyl-4-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
2-cyclohexyl-5-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}pyrimidine
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-11-{[2-(3-methoxyphenyl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-(2-methanesulfonylethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-3-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-2-(pyridin-3-yl)pyrimidin-4-ol
N-[4-({4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenyl]acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methylpentanamide
(3S,4R)-1-cyclobutanecarbonyl-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
8-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(4aR,7aS)-1-[2-(pyrrolidin-1-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}ethyl)acetamide
4-methyl-2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
[(3R,4R)-1-(1-benzothiophene-2-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(4-cyano-2-ethylphenyl)-3-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]urea
2-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}acetamide
4-(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)benzoic acid
1-(4-ethylpiperazin-1-yl)-3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}propan-1-one
N-ethyl-N-(2-hydroxyethyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,3-benzothiazole-6-carboxamide
2-{9-[4-(dimethylamino)benzoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-[(3R,4S)-4-cyclopropyl-1-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
1-(4-methoxy-3-methylbenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-{[2-(azepan-1-yl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)propanamide
methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})(quinoxalin-6-ylmethyl)amine
7-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
N-cyclohexyl-7-(pyridine-4-amido)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
(2-methylpropyl)[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
2-{2-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]propanamide
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-amine
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethan-1-one
4-(4-{[3-(1H-indazol-1-yl)propyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-({1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)cyclobutanecarboxamide
(2S,4S)-4-amino-1-(4-chloro-3-fluorobenzoyl)-N,N-diethylpyrrolidine-2-carboxamide
(1s,4s)-N1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}cyclohexane-1,4-diamine
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
(3S,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-methoxypiperidin-4-amine
3-{[(4-chloro-2-methoxy-5-methylphenyl)carbamoyl](methyl)amino}-N-methylpropanamide
4-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)phenyl]methyl}morpholine
5-(piperidine-1-carbonyl)-2-[3-(trifluoromethoxy)phenyl]pyridine
(1S,2R)-N1-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-N2-propylcyclohexane-1,2-dicarboxamide