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1-(2-ethylphenyl)-4-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazine
N,N-diethyl-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-3-carboxamide
(2S,4S)-N-ethyl-1-(3-methylbenzoyl)-4-[3-(methylsulfanyl)propanamido]pyrrolidine-2-carboxamide
N-cyclopentyl-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(2-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}ethyl)-1,3-oxazinan-2-one
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea
4-benzyl-3-ethyl-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-1,4-diazepan-5-one
(3R,4S)-4-cyclopropyl-1-{[2-methyl-5-(3-methyl-1,2-oxazol-5-yl)thiophen-3-yl]sulfonyl}pyrrolidin-3-amine
(3R,4S)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-4-(4-methoxyphenyl)pyrrolidin-3-amine
7-(cyclobutylmethyl)-2-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
1-ethyl-N-methyl-3-(propan-2-yl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
2-ethyl-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyrimidine-5-carboxamide
1-cyclopropanecarbonyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
4-[4-({2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}amino)piperidin-1-yl]-N,N-dimethylbenzamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)acetamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-3-azaspiro[5.5]undecan-9-amine
N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)propanamide
N-[2-(4-chlorophenyl)ethyl]-2-[(pyridin-2-ylmethyl)amino]acetamide
N-methyl-2-(1-{[(1-methyl-1H-indazol-3-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-4-carboxamide
1-[2-methoxy-4-(piperidin-1-ylmethyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
1-[4-({4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
(2R,3S,6R)-3-phenyl-5-(quinolin-5-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{3-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-5-ethyl-1,3,4-oxadiazol-2-amine
N-{4-[2-methyl-4-(3-methylphenyl)-5-oxopiperazine-1-carbonyl]phenyl}acetamide
2-{4-[4-(ethylcarbamoyl)pyridin-2-yl]phenyl}acetic acid
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4-(1H-pyrazol-3-yl)benzamide
({5-[1-(2-chloro-5-methylbenzoyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(1S,5R)-6-(dimethyl-1,3-oxazole-5-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
5-[bis(prop-2-en-1-yl)amino]-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrrolidin-2-one
1-[2-(4-fluorophenyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}ethoxy)ethan-1-ol
1,5-dimethyl-4-{6-oxo-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-8-yl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-[2-(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}morpholin-2-yl)ethyl]methanesulfonamide
5-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-{4-[2-(3-methylphenyl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}pentan-1-ol
7-(4-chlorophenyl)-2-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[(3-{[4-(morpholin-4-yl)butan-2-yl]carbamoyl}phenyl)amino]acetic acid
1-{[3-(3,3-diethylpyrrolidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-3-ol
N-[2-(2-chlorophenoxy)ethyl]-1-(pyridine-3-carbonyl)piperidin-4-amine
2-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-1-methyl-1H-indole
2-(3-methyl-1,2-oxazol-5-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-methylpiperazine-2-carboxylic acid
methyl({[1-(propan-2-yl)-1H-imidazol-2-yl]methyl})[3-(1H-pyrazol-1-yl)propyl]amine
4-(4-fluorophenyl)-1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,6-tetrahydropyridine
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one