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1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-phenylethan-1-one
(1S,5R)-3-[(3-chloro-1H-indol-2-yl)methyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1H-indole
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)acetamide
methyl 3-(2-chlorobenzamido)-6-[(3-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
3-{2-[1-(4-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}oxolan-2-one
(3aR,6aS)-2-(cyclopropylmethyl)-1-oxo-5-(pyrrolidine-1-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(5-acetylthiophen-3-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
(1H-imidazol-4-ylmethyl)({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
2-(azepan-1-yl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]acetamide
(1S,5S,6S,7R)-3-cyclohexyl-6-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-cyclopentyl-4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]acetamide
2-(2-{1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
3-{[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}propan-1-ol
5-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-2-carbonitrile
ethyl 4-[(4-chlorophenyl)methyl]-1-(3-methoxybenzoyl)piperidine-4-carboxylate
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-methylphenoxy)piperidine
methyl[(2-methyl-1,3-oxazol-4-yl)methyl][1-(pyridin-2-yl)propyl]amine
6-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazin-1-yl)pyrimidine-2,4-diamine
2-[2-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
3-[5-(5-oxo-5-phenylpentanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-cyclopentyl-4-(4-{[(5-methylfuran-2-yl)methyl]amino}piperidin-1-yl)benzamide
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
(2S,4R)-1-[(2-chlorophenyl)methyl]-N,N-diethyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-benzyl-3-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(4-chloro-3-methylphenyl)-2-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)acetamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
4-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
[(3R,5R)-5-[(dimethylamino)methyl]-1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl]methanol
5-methoxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-indazole-3-carboxamide
1-[(3,5-dichloro-2-hydroxyphenyl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(furan-3-carbonyl)pyrrolidin-3-yl]methanol
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N-cyclopropyl-1-{1-[4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}piperidine-3-carboxamide
2-(3-methoxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
N-[(3-methoxyphenyl)methyl]-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenylbenzamide
1-{9-[(3-fluorophenyl)methyl]-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl}-2-(methylsulfanyl)ethan-1-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(3S,4R)-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-4-propylpyrrolidin-3-yl]acetamide
4-benzyl-1-(2,4-dimethylpyrimidine-5-carbonyl)-3-ethyl-1,4-diazepan-5-one