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N-[(3-methylphenyl)methyl]-N-(propan-2-yl)pyridine-2-carboxamide
4-methyl-1-{2-oxo-2-[4-(pyridin-3-yl)piperazin-1-yl]ethyl}-1,2-dihydroquinolin-2-one
(3S,4R)-4-(hydroxymethyl)-1-(2-phenylquinolin-4-yl)piperidin-3-ol
9-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-8-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(2-{3-[1-(dimethylamino)ethyl]phenyl}-1H-imidazol-1-yl)methyl]benzoic acid
3-{1-[2-(morpholin-4-yl)benzoyl]piperidin-4-yl}phenol
dimethyl[1-(4-{1-[(3-methylpyridin-4-yl)methyl]-1H-imidazol-2-yl}phenyl)ethyl]amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
ethyl 1-[(4-hydroxyphenyl)methyl]-4-(2-phenylethyl)piperidine-4-carboxylate
3-[(4-methyl-6-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}pyrimidin-2-yl)amino]phenol
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
N-(4-methoxy-2-methylphenyl)-3-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
N-benzyl-1-{2-[3-(3-methoxyphenyl)propanamido]ethyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-imidazol-2-yl}pyridine
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(pyridin-3-yl)piperazine
4-[4-(pyridin-4-yl)pyrimidin-2-yl]-1λ6-thiomorpholine-1,1-dione
5-{[1-(hydroxymethyl)cyclobutyl]methyl}-11-methyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
3-({5-[1-(3,4-difluorophenyl)-1H-imidazol-2-yl]furan-2-yl}sulfanyl)-4-methyl-4H-1,2,4-triazole
1-(3-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}benzoyl)piperidine
N-cyclopropyl-3-{[(2S)-1-hydroxy-3-phenylpropan-2-yl]sulfamoyl}benzamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(6-methylpyridin-2-yl)methyl]propanamide
6-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
3-(1H-1,2,3-benzotriazol-5-yl)-1-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)urea
(4aR,8aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-[2-(4-fluorophenyl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]quinoline
1-cyclopentyl-4-({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)piperazin-2-one
3-amino-3-(3,4-dimethoxyphenyl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
3-{4-[(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-1H-pyrazol-1-yl}propanoic acid
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-4-(2-oxopiperidin-1-yl)butanamide
(4aR,7aS)-4-[2-(3-hydroxyphenyl)acetyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-(cyclopropylmethyl)-N,N-dimethyl-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-sulfonamide
3-{[3-(dimethylamino)-1-phenylpropyl]carbamoyl}benzoic acid
(1R,5S)-6-methyl-3-(1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(5-ethylpyridin-2-yl)methyl]-6-methoxy-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-(pyridine-2-carbonyl)piperidin-4-amine
2-(2-aminoethyl)-N-[3-(dimethylamino)propyl]-N,5,6-trimethylthieno[2,3-d]pyrimidin-4-amine
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
[(4-fluorophenyl)methyl](methyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
9-hydroxy-3-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
9-[(5-hydroxy-2-methoxyphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N3-methyl-4-oxo-1-(3-phenylpropyl)-N5-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-1,2-oxazolidine
4-(3-hydroxy-3-methylbutyl)-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
6-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-phenyl-5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]pyrimidin-2-amine
2-(4-chlorophenoxy)-1-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethan-1-one
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-1,4-dioxane-2-carboxamide