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N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
5-(3-chlorophenyl)-N-methyl-N-(quinolin-5-ylmethyl)-1,2,4-triazin-3-amine
3-butyl-4-ethyl-1-{2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(3-methoxypropyl)piperidin-1-yl]-2-phenylethan-1-one
N-[(3-hydroxypyrrolidin-3-yl)methyl]-4-(piperidin-1-yl)benzamide
(2-{2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2,6-dihydroxy-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
2-[(2S,3R)-2-amino-3-hydroxybutanoyl]-N-cyclobutyl-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-2-(trifluoromethyl)morpholine
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-2,5-dimethylfuran-3-carboxamide
4-benzyl-3-[1-(5-fluoropyridine-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetate
2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazole
5-cyclopropanecarbonyl-1'-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2,1,3-benzoxadiazole
N,N-dimethyl-3-[3-(2-phenylacetyl)piperidin-1-yl]propane-1-sulfonamide
1-{3-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenyl}ethan-1-one
6-(2-chlorophenyl)-N,N-dimethyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-fluoro-6-methoxybenzamide
5-({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1,2-oxazol-5-yl}methoxy)-2-methyl-1,3-benzothiazole
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,3-dihydro-1-benzofuran-5-carboxamide
5-[(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)carbamoyl]-1H-imidazole-4-carboxylic acid
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
4-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}-3-methylpiperazin-2-one
N-methyl-3-(propan-2-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1,2-oxazole-5-carboxamide
4-[(4-fluorophenyl)sulfanyl]-1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidine
1-{[1-(3-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyridin-2-one
N-[(4-fluorophenyl)methyl]-N-(2-hydroxyethyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-(4-chlorophenyl)-N-(2-methanesulfonylethyl)-3-phenylpropanamide
2-(2,6-dimethoxyphenyl)-5-fluoro-4-methoxypyrimidine
3-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
2-chloro-N-[1-(1-methylpiperidin-4-yl)-1H-pyrazol-5-yl]benzamide
(2S,4R)-1-benzyl-4-{[(2,6-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-[2-(azepan-1-ylmethyl)phenyl]-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
3-{[(2,5-dimethylphenyl)methyl]amino}-N-[2-(1H-imidazol-1-yl)ethyl]-5-(pyrrolidine-1-sulfonyl)benzamide
2-(2-ethoxyphenyl)-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R,5S)-1-benzyl-N-(2,3-dihydro-1H-inden-5-yl)-5-[3-(dimethylamino)pyrrolidine-1-carbonyl]piperidine-3-carboxamide
4-cyano-N-[(3R,4S)-4-cyclopropyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]oxane-4-carboxamide
methyl 3-(cyclobutylmethoxy)-5-[(1-methylpiperidin-3-yl)carbamoyl]benzoate
2-[(5-hydroxy-6-methyl-1,2,4-triazin-3-yl)sulfanyl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]acetamide
4-(1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)morpholine
4-benzyl-1-(2,5-dimethylpyrimidin-4-yl)-3-ethyl-1,4-diazepan-5-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylpropanamide
1-cyclobutyl-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
N-ethyl-N-(1-hydroxypropan-2-yl)-2-phenylbenzamide
N-[3-(1H-imidazol-1-yl)propyl]-1-methyl-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(3-fluorophenyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
1-[4-({[2-(4-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
N-[(1R)-1-(3-methoxyphenyl)ethyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine