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4-hydroxy-N-[2-(pyridin-2-yl)ethyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
ethyl 5-({1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}carbamoyl)-1H-imidazole-4-carboxylate
2-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
1-{4-[2-({[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl)amino}methyl)-8-methylquinazolin-4-yl]-1,4-diazepan-1-yl}ethan-1-one
N,N-dimethyl-1-[(6-methylquinolin-5-yl)methyl]azepan-4-amine
2-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
(1R,7S)-3-(4-fluorophenyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-{2-[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-3-carboxamide
2-amino-2-methyl-1-(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)propan-1-one
methyl 2-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-1,3-oxazole-4-carboxylate
2-[4-(1H-imidazol-1-yl)phenyl]-N-methylacetamide
2-({4-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}sulfanyl)ethan-1-ol
3-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
N-(4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)acetamide
2-(2-{[(4aS,7aR)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}phenoxy)acetic acid
4-{4-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}thiomorpholine
2-chloro-N-methyl-5-[1-(3-methylbutyl)-1H-pyrazol-4-yl]benzamide
[3-(2-methylpropyl)-1-(thiophen-2-ylmethyl)piperidin-3-yl]methanol
1-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-(3-chlorophenyl)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-[(4-ethoxyphenyl)methyl]-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}cyclopropanamine
(3aR,6aS)-2-(cyclopropylmethyl)-5-(2-methylfuran-3-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-4-(dimethylamino)-1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidine-2-carboxylic acid
(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1,2,3,6-tetrahydropyridine
6-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]quinoline
2-(diethylamino)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
5-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
1-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
6-({4-[2-(morpholin-4-yl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}methyl)-1H-indole
1-ethyl-4,6-dimethyl-3-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
2-[2-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyrimidine
1-methyl-N-[(3-methylpyridin-2-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-methyl-7-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
9-(2-hydroxyethyl)-1-methyl-4-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-(morpholin-4-yl)butanamide
7-(2,2-dimethylpropyl)-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
3-methyl-2-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]pyridine
N-(1-ethyl-1H-indazol-3-yl)-2-(4-phenyl-1H-imidazol-1-yl)acetamide
methyl (2S)-2-{[1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-3-yl]formamido}-2-phenylacetate
3-chloro-N-(2-methoxyethyl)-4-{[1-(thiophen-3-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(1-{1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
1-(2-{[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,4-triazole
N,1-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl]-3-(methylsulfanyl)propanamide
1-[(4-methoxyphenyl)methyl]-4-(4-phenylbutanoyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]benzene-1-sulfonamide