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3-methyl-2-{5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl}pyridine
8-[1-(1-methylpiperidin-4-yl)-4-phenyl-1H-imidazol-5-yl]quinoline
N-[2-(2-oxopiperidin-1-yl)ethyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
[(2S)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-2-yl]methanol
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(5-methylpyrazin-2-yl)methyl]pyridin-2-amine
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-4-(propan-2-yl)piperazine
8-[3-(4-methoxyphenyl)benzoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-(5-chloro-2-methoxyphenyl)-2-[methyl(pyridin-2-ylmethyl)amino]acetic acid
N-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
8-(2-aminopyrimidin-4-yl)-3-{2-[methyl(2-phenylethyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
5-cyclopropanecarbonyl-1'-(1-methyl-1H-imidazole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyrazin-2-amine
1-(2-aminopyrimidin-4-yl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
6-[(3-methoxyphenyl)methoxy]-4-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-1-(2-phenylethyl)-1,4-diazepan-2-one
2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-4-methyl-1H-1,3-benzodiazole
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-(pyridin-3-yl)propanamide
5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazin-2-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)propanamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
3-cyclobutyl-4-(2-phenylethyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-butyl-1'-(2-methyl-1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(4-chloro-2-methylbenzoyl)-3-ethylpiperazine
(3S,4R)-3-ethyl-4-methyl-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-ol
1-(2-ethoxyethyl)-5-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
7-methoxy-4-methyl-3-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2H-chromen-2-one
N-phenyl-5-(propane-2-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-amino-6-(2-methylpropyl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]pyrimidine-4-carboxamide
(1S,5R)-6-benzyl-3-(5-ethyl-2-methylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[(3-phenylphenyl)methyl]piperidin-4-ol
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
2-(naphthalen-1-yl)-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
4-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
N,N-diethyl-1-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]piperidine-3-carboxamide
(4S,6R)-6-methyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-2-sulfanylidene-1,3-diazinane-4-carboxamide
1-(piperidine-1-sulfonyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-diazepane
2-(2H-1,2,3-benzotriazol-2-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
4-methyl-5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrazine
5-(morpholin-4-ylmethyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]furan-3-carboxamide
N-(2-methoxy-5-methylphenyl)-2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]acetamide
4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-sulfonyl]-N-[(2R)-oxolan-2-ylmethyl]benzamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-3-carboxylic acid
4-ethyl-3-[1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one