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(3-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
1-(4-methoxyphenyl)-3-methyl-4-[2-(thiophen-3-yl)acetyl]piperazin-2-one
N-ethyl-2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]pyridine-4-carboxamide
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}but-3-en-1-one
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-5-(morpholin-4-ylmethyl)-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-3-(1H-imidazol-1-ylmethyl)piperidine
1-methyl-4-[(6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridin-3-yl)methyl]piperazine
{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
6-[({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)methyl]-1,4-oxazepan-6-ol
(1R,9S)-5-amino-3-[2-(2-hydroxyethoxy)phenyl]-13-methyl-6,13-diazatricyclo[7.3.1.02,7]trideca-2,4,6-triene-4-carbonitrile
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)cyclobutanecarboxamide
7-(1-benzothiophen-3-yl)-4-(furan-2-carbonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-ethyl-6-methyl-5-{2-oxo-2-[2-(trifluoromethyl)morpholin-4-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-[3-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
4-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]-2-(trifluoromethyl)morpholine
2-(6-methoxy-1H-indol-2-yl)pyridin-4-amine
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-2-(4-propanoylphenoxy)acetamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(4-methyl-1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[(3-methoxyphenyl)methyl]piperidine-3-carboxamide
2-chloro-N-[(1-ethylpiperidin-3-yl)methyl]pyridine-4-carboxamide
(3S,7S,8aS)-7-{[(2-fluorophenyl)methyl]amino}-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
7-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
(3S,4S)-4-(dimethylamino)-1-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}pyrrolidin-3-ol
N-[(4-hydroxyphenyl)methyl]-2,7-dioxo-N-(pyridin-3-ylmethyl)-1,3-diazepane-4-carboxamide
2-[1-ethyl-2,4-dioxo-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
(3R,4R)-1-(4-methoxybenzoyl)-4-{[(5-methylpyrazin-2-yl)methyl]amino}pyrrolidin-3-ol
4-{2-methyl-6-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
1-{3-[(butan-2-yl)amino]propyl}piperidin-4-ol
(3R,4R)-4-(hydroxymethyl)-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]piperidin-3-ol
1-{[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}-1,4-diazepan-5-one
3-(4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-5-chloro-1-methyl-1H-pyrazol-3-yl)-5-methyl-1,2-oxazole
5-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)piperidin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(1H-indol-3-yl)-N-methylacetamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazine
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-3-yl}propan-1-one
(2S,4S)-1-(3,3-dimethylbutanoyl)-4-(2,5-dimethylfuran-3-amido)-N-ethylpyrrolidine-2-carboxamide
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(thiophen-3-ylmethyl)benzamide
3-{[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
1-methyl-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
3-[4-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]prop-2-yn-1-ol
N-(1-fluoro-3-phenylpropan-2-yl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
3-{methyl[2-(methylsulfanyl)ethyl]sulfamoyl}-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
(1-{[(2-butoxy-3-methoxyphenyl)methyl]amino}cyclopentyl)methanol
N-cyclopentyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
ethyl 5-(2-hydroxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine