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(4aS,8aS)-2-[5-(piperidin-1-ylmethyl)pyridin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
5-(3,4-dimethoxyphenyl)-2,3-dihydro-1,3-benzoxazol-2-one
(2S)-2-hydroxy-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-phenylpropanamide
4-[2-(dimethylamino)phenyl]-5H,6H,7H-cyclopenta[d]pyrimidin-2-amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
1-ethyl-5-oxo-N-[2-(2-phenoxyphenyl)ethyl]pyrrolidine-3-carboxamide
2-methoxy-1-{4-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]piperidin-1-yl}ethan-1-one
7-fluoro-3-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-1-(pyridin-3-ylmethyl)-1,2-dihydroquinolin-2-one
4-{3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}phenol
2-[(4aR,7aS)-4-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
4-[(1E)-1-phenylprop-1-en-2-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2-methoxyethyl)-3-(2-methylpropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopentanecarbonyl-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3S,4S)-4-cyclopropyl-1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}pyrrolidine-3-carboxylic acid
(1R,7S)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(2-{3-[(2,6-dichlorophenyl)methyl]-1-ethyl-1H-1,2,4-triazol-5-yl}ethyl)methanesulfonamide
5-{[benzyl(methyl)amino]methyl}-N-[2-(1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
[(3-chloro-5-fluoro-4-methoxyphenyl)methyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
3-(2-methoxyphenyl)-N-(oxolan-3-yl)propanamide
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
(2S,5R)-1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,5-dimethylpiperazine
(2S,4R)-4-[(adamantan-2-yl)amino]-1-benzyl-N-(propan-2-yl)pyrrolidine-2-carboxamide
dimethyl({[1-(quinoline-6-carbonyl)piperidin-3-yl]methyl}sulfamoyl)amine
N-{[1-(4-cyano-1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}-4-fluorobenzamide
7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-fluorophenyl)-4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperazine
methyl 2-(azepane-1-sulfonyl)-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl 1-{7-chloro-3-[(cyclopentylamino)methyl]quinolin-2-yl}piperidine-3-carboxylate
1-(5-chloronaphthalene-1-carbonyl)-4-(4-methoxybutyl)piperazine
8-chloro-2-(oxolane-3-carbonyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-methyl-4-(4-methyl-1,4-diazepan-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propane-1,2-diol
5-ethyl-2,3-dimethyl-N-[1-(6-methylpyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-methyl-5-[5-(1-methyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]-2-(pyridin-2-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
3-{[1-(3,4-dimethylbenzoyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopropyl-5-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
N-[2-(1H-indol-3-yl)ethyl]-1-methyl-N-(pyridin-3-ylmethyl)azepane-2-carboxamide
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(3-oxopiperazin-1-yl)acetamide
1-(4-fluorophenyl)-4-(3-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
4-methoxy-N-(2-methoxyethyl)-2-({1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}oxy)benzamide
3-cyclopropyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2-oxazole
(3R,4S)-3,4-dimethyl-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-4-ol
1-[2-methoxy-1-(pyridin-2-yl)ethyl]-3-(5-phenyl-1,3,4-thiadiazol-2-yl)urea
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(furan-2-yl)propan-1-one
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one