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6-[(2-fluorophenyl)methoxy]-4-(1-methylpiperidin-4-yl)-1-(2-methylpropyl)-1,4-diazepan-2-one
(2R,3R,6R)-5-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1S,5R)-3-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-[2-(3,4-dimethylphenyl)ethyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
methyl 3-benzamido-5-{[1-(methylsulfanyl)propan-2-yl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-cyclopropaneamido-N,4-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
(2S)-2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]-3-(pyridin-4-yl)propanoic acid
2-cyclohexyl-6-[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
5-{2-[(2-methoxyethyl)amino]ethyl}-1-(3-methylbutyl)pyrrolidin-2-one
6-hydroxy-N-[4-(3-methoxyphenoxy)phenyl]-1,4-oxazepane-4-carboxamide
[5-chloro-7-(6-phenylpyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N,N-dimethyl-3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-sulfonamide
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-[4-(trifluoromethoxy)phenyl]urea
N-[(2-methoxyphenyl)methyl]-4-(piperidin-3-ylmethyl)benzamide
2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-4-carboxamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-3-ol
8-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N4-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3-ethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[(1-methylpiperidin-4-yl)amino]methyl}hepta-1,6-dien-4-ol
4-cyclobutaneamido-N-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
5-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1-[(1-methylpyrrolidin-3-yl)methyl]-4-phenyl-1H-imidazole
1-ethyl-3-{3-[2-(4-methoxyphenyl)ethyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
(3aR,6aR)-2-cyclobutanecarbonyl-5-(4-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-({[3-(pyridin-4-yl)propyl]amino}methyl)-1,4-oxazepan-6-ol
2-{2-[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-({5-[(2S)-azetidine-2-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-ethoxypiperidine
2-[4-(furan-3-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-1-(piperidin-1-yl)ethan-1-one
2-methoxy-3-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyrazine
4-({6-[6-(benzyloxy)pyridin-3-yl]pyridin-3-yl}methyl)morpholine
[(1-cyclohexylpiperidin-3-yl)methyl][(3,4-dimethoxyphenyl)methyl](pyridin-3-ylmethyl)amine
1-(2,4-difluorophenyl)-3-methyl-5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazole
(1H-imidazol-2-ylmethyl)(methyl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(3-methylpyridin-2-yl)propan-2-yl]propanamide
2-fluoro-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-5-sulfamoylbenzamide
4-{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidin-4-yl}pyridine
1-(cyclopropylmethyl)-N-ethyl-5-(1H-indol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(5-{3-[1-(dimethylamino)ethyl]phenyl}-2-methoxyphenyl)methanol
3-hydroxy-1-(2-phenylethyl)-3-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)piperidin-2-one
2-chloro-N-[(3-hydroxypyrrolidin-3-yl)methyl]-5-(trifluoromethyl)benzamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)pyridine-2-carboxamide
7-(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-N-ethyl-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(4-fluorophenyl)methyl]-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
3-{[(4-hydroxybutyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
9-(cyclopropylmethyl)-4-(2-ethoxyacetyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-cyclopropyl-1-[1-(quinolin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-(4-chlorophenyl)-N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
N-(2-methyl-1-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)methanesulfonamide