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4-[2-(cyclohex-1-en-1-yl)acetyl]-6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
2-(2,4-dichlorophenoxy)-N-[2-(oxan-3-yl)ethyl]acetamide
2,3,5-trimethyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-methyl-2-(6-methylpyridin-2-yl)-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
1-[(4-fluorophenyl)methyl]-4-(5-methyl-1,2-oxazole-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
[(3S,4S)-4-(hydroxymethyl)-1-(trimethylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
2-(2-methyl-1,3-thiazol-4-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
3-({[2-(1H-imidazol-1-yl)phenyl]methyl}amino)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}cyclohex-1-ene-1-carboxamide
N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-acetyl-N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]piperidine-3-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
methyl (2S)-2-({[(2,4-dimethylphenyl)carbamoyl]methyl}amino)-2-phenylacetate
N-[3-(3-cyanopyridin-2-yl)phenyl]acetamide
3-(4-hydroxyphenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]propanamide
3-[2-(dimethylamino)ethyl]-8-[(3-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-(2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazine-1-carboxylate
N-{1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]pyrrolidin-3-yl}acetamide
3-{[8-(1,3-benzothiazol-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenol
4-(4-{[cyclopropyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-2-methylbutan-2-ol
5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-methyl-4-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)pyridin-2-yl]piperazine
2-methyl-8-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
3-methyl-7-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-(2-amino-4-methyl-6-{methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}pyrimidin-5-yl)propanoic acid
3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
2-cyclopropyl-4-hydroxy-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]pyrimidine-5-carboxamide
3-[2-(dimethylamino)ethyl]-3-ethyl-1-[2-(pyridin-2-ylmethoxy)phenyl]urea
4-{[1-(3,5-dimethyl-1H-indol-2-yl)-N-ethylformamido]methyl}benzoic acid
2-(4-methyl-6-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}pyrimidin-2-yl)phenol
(3aS,7aR)-2-[(5-ethylpyridin-2-yl)methyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-(4-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
N4,5-dimethyl-N4-(3-phenoxypropyl)pyrimidine-2,4-diamine
4-methoxy-6-(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)pyrimidine
9-ethyl-1-methyl-4-[(1-methyl-1H-indol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}-1-(pyrrolidin-1-yl)propan-1-one
(1S,4S)-2-(3-chlorophenyl)-5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(2S,4R)-4-{[(2-fluorophenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
N-[(2S)-pyrrolidin-2-ylmethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-3-methanesulfonamidopropanamide
2-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({[3-(trifluoromethoxy)phenyl]methyl})amine
N-(3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-2,5-dimethyl-1H-pyrrol-1-yl)acetamide
3-cyclopropyl-1-methyl-4-[5-(piperidin-1-ylmethyl)thiophen-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one