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5-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
methyl 5-{[(2-fluorophenyl)methyl]amino}-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]cyclopent-1-ene-1-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-(7-methyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylacetamide
2-{1-[(1-butylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
2-{2-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-oxoethyl}-4-phenyl-1,2-dihydrophthalazin-1-one
1-(5-methoxyfuran-2-carbonyl)-3-[2-(3-methoxyphenyl)ethyl]piperidine
2-methyl-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-cyclopropyl-9-[2-(1H-imidazol-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-cyclobutanecarbonyl-3-(3-phenylpropyl)piperidine-3-carboxylate
4-(1H-imidazol-2-yl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidine
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
4-{4-[1-(3-methylbutyl)-1H-pyrazol-4-yl]phenyl}morpholine
2-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
2-methyl-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
6-[methyl(1-methylpyrrolidin-3-yl)amino]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
1-cycloheptyl-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
3-(4-fluorophenoxymethyl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine
3-[(5-oxo-1,4-diazepan-1-yl)sulfonyl]-N-[(2S)-oxolan-2-ylmethyl]benzamide
3-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(6-methylpyrimidin-4-yl)piperidin-3-yl]propan-1-ol
4-(benzyloxy)-N-(5-carbamoyl-2-methylphenyl)piperidine-1-carboxamide
1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-oxopyrrolidine-3-carboxylic acid
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
1-[(1S)-1-cyclohexylethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-{[2-(adamantan-1-yl)-1,3-thiazol-4-yl]methyl}-1,4-oxazepane
2-{4-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]phenoxy}acetic acid
5-{3-[1-(3-methoxypropyl)-1H-pyrazol-3-yl]phenyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
4-(pyridin-2-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrimidin-2-amine
2-(dimethylamino)-2-(4-fluorophenyl)-N-[1-(hydroxymethyl)cyclopentyl]acetamide
1-{4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]phenyl}-3-ethylurea
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-{4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine
7-fluoro-3-[({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2-dihydroquinolin-2-one
3-fluoro-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-methoxybenzamide
3-(2-methoxyphenyl)-6-[3-(pyridine-2-carbonyl)piperidin-1-yl]pyridazine
(1S,6R)-9-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
N-(1,4-dioxan-2-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(2-chlorophenyl)-4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-2-one
N-[2-(4-chlorophenyl)ethyl]-2-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}acetamide
5-methanesulfonyl-1'-(pyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-ethoxy-2-{[3-(methoxymethyl)piperidin-1-yl]methyl}quinoline
5-[3-(3-hydroxy-3-methylbutyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-(methylsulfanyl)-3-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one