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5-[(2E)-2-methylbut-2-en-1-yl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-methyl-1-(4-{5-[2-(1-methylpiperidin-3-yl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)-1H-pyrazol-5-amine
2-(1H-indol-3-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1λ6-thiolane-1,1-dione
ethyl 2-{N-methyl-1-[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]formamido}acetate
3-[3-(propan-2-yloxy)phenyl]-1-[3-(pyridin-2-yl)propyl]urea
methyl 1-(benzylsulfamoyl)piperidine-2-carboxylate
N-methyl-4-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
3-[1-(4-chloro-2-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
2-methyl-5-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenol
4-[(3-fluorophenyl)methyl]-3-{2-oxo-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethyl}piperazin-2-one
5-chloro-2-(2-methyl-1,4-oxazepane-4-carbonyl)-3-phenyl-1H-indole
5-chloro-N-[2-(dimethylamino)ethyl]-N-methyl-3-phenyl-1H-indole-2-carboxamide
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidine
(2S,4S)-4-(4-{2-[(2-chlorophenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}thiomorpholine
N,N-dimethyl-3-({[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}sulfamoyl)benzamide
N-cyclopropyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}oxolane-2-carboxamide
4-(4-methoxy-2-methylphenyl)pyridin-2-amine
7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R)-1-[(1-{[1-(3-fluorobenzoyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-amine
2-(1,1-dioxo-1λ6-thiomorpholin-4-yl)-N-[1-(4-methylphenyl)ethyl]acetamide
4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-1,2-dihydroquinolin-2-one
(1H-imidazol-4-ylmethyl)[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
1-cyclopentyl-4-[({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]pyrrolidin-2-one
N-(2-methoxyethyl)-N-(naphthalen-1-ylmethyl)-2-(piperidin-4-yl)acetamide
3-[(1-phenylmethanesulfonylpyrrolidin-3-yl)methyl]benzamide
2-(pyridin-4-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]quinoline-4-carboxamide
1-{2-[3-(methanesulfonylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methyl-1H-indole
4-({2-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[(1S,5R)-3-[2-(1,2-benzoxazol-3-yl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-(3-cyclopropyl-1-propyl-1H-1,2,4-triazol-5-yl)-1,2-dihydroquinolin-2-one
7-(pyridin-3-yl)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}benzoic acid
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-({1-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
8-[(4-methoxyphenyl)methyl]-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
3-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1-phenylurea
(4R)-4,7,7-trimethyl-1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]-2-oxabicyclo[2.2.1]heptan-3-one
N'-(2-ethoxyphenyl)-N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)propanediamide
(4aS,7aR)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2-fluorophenyl)-N-(1,3-thiazol-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[2-(cyclohex-1-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
(2S,4S)-4-amino-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-N,N-diethylpyrrolidine-2-carboxamide
N-(pyridin-2-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine