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5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridin-2-amine
2-(3-hydroxypropyl)-8-[4-(trifluoromethyl)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
5-fluoro-2-[1-(pyridin-3-ylmethyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-ethyl-5-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}pyrimidin-2-amine
6-tert-butyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-chloro-5-acetamido-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
2-[(3-methylpiperidin-3-yl)methoxy]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
7-fluoro-N-(3-hydroxypropyl)-N-[(2-methoxyphenyl)methyl]-2-methylquinoline-4-carboxamide
5-ethyl-5-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[(5-phenyl-1H-pyrazol-3-yl)methyl]amine
4-(2,2-dimethyl-3-{4-[(3-methylphenyl)methyl]piperazin-1-yl}propyl)morpholine
1-ethyl-4-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
1-[1-(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[3-(morpholin-4-yl)propyl]benzamide
1-(oxolane-2-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-[(1S,2R)-2-(cyclooctylamino)cyclobutyl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetamide
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-phenyl-N-{1-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
1-[(5-ethylpyridin-2-yl)methyl]-4-{thieno[3,2-d]pyrimidin-4-yl}piperazine
2-ethyl-9-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
ethyl(oxolan-2-ylmethyl)(quinolin-4-ylmethyl)amine
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(4,5-dimethyl-1H-imidazol-1-yl)ethan-1-one
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
3-[2-(2-fluorophenyl)ethyl]-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
3-(2-methylphenyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-yl]methanol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(pyridine-3-carbonyl)piperidin-3-yl]piperazine
2-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
2-({[(3S,4R)-1-[(2,4-difluorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
(2S,4S)-4-(benzylamino)-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-{4-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-(oxan-4-yl)piperidine
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine
1-(furan-3-carbonyl)-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4-diazepane
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(1H-imidazol-1-yl)-N-methylbenzamide
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3-phenylpyrrolidin-3-ol
4-(2-methoxyacetyl)-N-[2-(methylsulfanyl)phenyl]-1,4-diazepane-1-carboxamide
N-[2-(1H-indol-3-yl)ethyl]-N-(pyridin-3-ylmethyl)oxane-4-carboxamide
7-[3-(4-methoxyphenyl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(5-chloro-2-fluorobenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-amino-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-6-(naphthalen-2-yl)pyridine-3-carbonitrile
5-methyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
7-[(2-fluorophenyl)methyl]-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decane
2-(propan-2-yl)-5-[3-(pyridine-3-carbonyl)piperidine-1-carbonyl]-1,3-benzoxazole
1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one