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3-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-N-(furan-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]pyridine-4-carboxamide
2-phenyl-N-(propan-2-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
2-(3-methyl-4-{[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
1-(1-cyclohexylpiperidine-4-carbonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
5,5-dimethyl-3-{2-oxo-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}imidazolidine-2,4-dione
N-{2-oxo-2-[3-(2-phenylacetyl)piperidin-1-yl]ethyl}benzamide
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
[(3-chloro-5-fluoro-4-methoxyphenyl)methyl](furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amine
N-cyclopropyl-4-methoxy-2-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
2,5-dimethyl-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-1,3-thiazole-4-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]propanamide
N-(2-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
N-[1-(1-benzylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxybenzamide
1-{2-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
2-methoxy-3-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]methyl}-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethan-1-amine
4-[(furan-2-ylmethyl)amino]-5-methyl-N-[2-(propan-2-yloxy)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-phenyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
[(3R,4S)-1-[(4-chloro-3-fluorophenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-(3,4-dimethoxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(4-methoxy-2-methylphenyl)-3-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-yl)propanamide
2-(3-methoxyphenyl)-3-[(4-methylpiperazin-1-yl)methyl]-7-(methylsulfanyl)quinoline
1-ethyl-5-{[(3-fluoro-4-methylphenyl)methyl]amino}-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-({4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)benzonitrile
2-cyclopropyl-N-[(3R,4S)-1-[2-(methylcarbamoyl)ethyl]-4-propylpyrrolidin-3-yl]pyrimidine-5-carboxamide
N-[(2R,3R)-2-ethoxy-1'-[(3-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
2-[1-(propan-2-yl)piperidin-4-yl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]acetamide
3-(1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-methyl-1H-pyrrole-3-carbonyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-4-methylbenzamide
1-[2-({[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}(methyl)amino)ethyl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
6-methoxy-3-methyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1-benzofuran-2-carboxamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-(piperidin-4-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1S,5R)-3-[(2-ethylphenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-{2,7-diazaspiro[4.5]decane-7-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N-[2-(azepan-1-yl)ethyl]-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
9-[(3-fluoro-2-methoxyphenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(4-propanoylphenoxy)acetamide
N-[(3-methoxyphenyl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-[3-(furan-2-yl)propyl]-1-methyl-1H-indole-6-carboxamide
3,4,7-trimethyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-indole-2-carboxamide
2-(3-acetamidophenyl)-6-methylpyridine-3-carboxamide
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-3-(pyridin-3-yl)propan-1-one
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-(2-methoxyethyl)-1-[(4-oxo-4H-chromen-3-yl)methyl]pyrrolidine-2-carboxamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-[4-(propan-2-yl)morpholin-2-yl]acetamide