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2-(dimethylamino)-2-(2-fluorophenyl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
1-[(2-ethylpyrimidin-4-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
4-{6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-4-yl}morpholine
7-cyclopentyl-2-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
(4aS,8aR)-1-(2-aminoethyl)-6-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-(3-acetylphenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[({3-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)(methyl)amino]propanamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
(2S,4R)-4-[(adamantan-2-yl)amino]-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
6-methyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-[3-fluoro-5-(trifluoromethyl)phenyl]-N,N-dimethylbenzamide
3-(3,4-difluorophenyl)-N-(furan-2-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(1,3-thiazol-2-yl)piperidine-3-carboxamide
4-methyl-2-{2-oxo-2-[4-(pyridin-3-yl)piperazin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
4,5-dimethyl-6-(1H-pyrazol-3-yl)-2-(trifluoromethyl)pyrimidine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
2-cyclohexyl-6-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,3-benzoxazole
[(1-cyclopentylpiperidin-4-yl)methyl][(2-ethoxyphenyl)methyl](pyridin-3-ylmethyl)amine
4-phenyl-1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-ol
3-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
(1,4-dioxan-2-ylmethyl)({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-[2-fluoro-5-({[1-(4-methoxyphenyl)propyl](methyl)carbamoyl}amino)phenyl]acetamide
N-(furan-2-ylmethyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
8-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
ethyl 2-[(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)amino]-1H-imidazole-5-carboxylate
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-6-(3-methoxyphenyl)pyridine-3-carbonitrile
2-{2-[6-amino-5-cyano-4-(3,5-dimethyl-1H-pyrazol-4-yl)pyridin-2-yl]phenoxy}acetamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidine-2,4-diamine
3-{2-[5-(3-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
4-{[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl](pyridin-3-yl)methyl}morpholine
3-hydroxy-3-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
2-[1-(1H-indole-5-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
N-[7-methoxy-4-(1-methyl-1H-indol-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]butanamide
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
(1S,5R)-6-benzyl-3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 3-methyl-4-{[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]amino}benzoate
[(3-fluoro-2-methoxyphenyl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
N7-(6-chloropyridin-3-yl)-2,N3,N3-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3,7-dicarboxamide
dimethyl(3-{2-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
3-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-1-ium-1-olate
dimethyl({4-methyl-5-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]azocane
1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(hydroxymethyl)azepan-4-ol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{4-[2-(dimethylamino)ethoxy]-1-(3-fluorophenyl)-1H-indazol-3-yl}oxolane-3-carboxamide
N-[2-(dimethylamino)-1-phenylethyl]-1-ethyl-N-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-{4-methyl-6-[4-(oxolan-2-ylmethyl)piperazin-1-yl]pyrimidin-2-yl}phenol