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2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-diethylacetamide
[(5-ethylfuran-2-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
3-(1-methanesulfonylpiperidin-4-yl)-1-(2-methylquinolin-8-yl)urea
1-benzyl-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(2-methylpropanesulfonyl)-1H-imidazole
methyl 8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amine
N-(2-hydroxyethyl)-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
4-ethyl-3-(1-ethyl-1H-pyrazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(4-fluorophenoxy)piperidine
1-{4-[(dipropylamino)methyl]benzoyl}-2-methyl-1,4-diazepan-5-one
3-[3-(4-chlorobenzoyl)piperidine-1-carbonyl]-2H-chromen-2-one
2-[1-(3-methylbut-2-en-1-yl)-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl]ethan-1-ol
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazole
4-hydroxy-1-[4-(trifluoromethyl)pyridin-2-yl]piperidine-4-carboxylic acid
2-[2-(4-methoxy-3,5-dimethylphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-hydroxy-5-methylbenzoyl)pyrrolidine-3-carboxylic acid
6-({[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
8-[(3-chlorophenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2-chlorophenyl)-3-[2-(methylsulfanyl)ethyl]-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
5-({[(4-hydroxy-6-methylquinolin-2-yl)methyl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-indole-7-carboxamide
N-butyl-N-(furan-2-ylmethyl)pyrrolidine-3-carboxamide
2-methyl-5-[4-(thiophen-3-ylmethyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,2,6,6-tetramethylpiperidin-4-amine
(1S,5R)-6-(cyclopropylmethyl)-3-[2-(4-methoxyphenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-amino-1-[(2-hydroxyphenyl)methyl]pyrrolidine-3-carboxylic acid
5-({2-[5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,4-triazole
N-{2-[5-(2,3-dimethyl-1H-indol-7-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N-ethyl-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-amido]piperidine-1-carboxamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(4-methylpyridin-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[(2-ethyl-1-benzofuran-3-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-[(3R,4S)-3-cyclobutaneamido-4-cyclopropylpyrrolidin-1-yl]-6-methylpyridine-3-carboxylic acid
(1S,5R)-3-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(5-methylfuran-2-yl)-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
1-benzyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methoxy-4-{2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyridine-3-carbonitrile
2-hydroxy-N-methyl-N-[(5-methylfuran-2-yl)methyl]-5-(1H-pyrrol-1-yl)benzamide
1-(4-{[3-(dimethylamino)butyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
2-({[(1R,2S)-2-hydroxycyclohexyl](methyl)amino}methyl)-3,5-dimethoxybenzoic acid
3-(4-methyl-1,3-thiazol-5-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}propanamide
3-[1-(oxolane-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(3-methylthiophen-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
1-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea