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(4aS,8aR)-6-(1H-imidazol-4-ylmethyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-(1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)pyrimidine
N-(pyridin-2-ylmethyl)-2-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}acetamide
[1-({4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-3-yl]methanol
[(3-{[1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
3-methoxy-1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-1,2-dihydropyridin-2-one
2-(4-{4-[4-(pyridin-3-yloxy)piperidin-1-yl]piperidin-1-yl}benzoyl)-1,2,3,4-tetrahydroisoquinoline
(2S,4R)-4-amino-1-(2-methoxypyridine-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(4-hydroxypiperidin-1-yl)ethyl]-4-(piperidin-3-yl)benzamide
2-chloro-4-[4-(morpholin-4-yl)phenyl]benzamide
2-(5,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
(2S)-N-(5-acetyl-2-methoxyphenyl)-2-(piperidine-1-carbonyl)pyrrolidine-1-carboxamide
2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylacetamide
4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-6-ethyl-1,2-dihydropyridin-2-one
2-methyl-3-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
2-{4-[(3-hydroxypyrrolidin-3-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
8-acetyl-2-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(3-acetamido-4-methoxyphenyl)-4-(2-ethoxyethyl)piperazine-1-carboxamide
N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(oxan-2-ylmethyl)acetamide
4-[3-cyclopropyl-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
6-{[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}phenyl)methyl]pyrrolidin-2-one
2-{4-[(3-fluorophenyl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
2-hydroxy-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethylpropanamide
ethyl 1-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}piperidine-4-carboxylate
N-[(3R,4S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
(1S,4S)-5-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(1S,3R)-N1-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
1-(5-acetylpyridin-2-yl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
5-{[2-(2-chlorophenyl)ethyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-2,7,8-trimethylquinoline-4-carboxamide
(4aR,8aR)-7-[(3-fluorophenyl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
6-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
ethyl 2-({3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}amino)acetate
1-[(3-fluorophenyl)methyl]-4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazine
(3S)-4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-ethylmorpholine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
3-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1H-pyrazol-5-amine
1-methyl-5-{2-[2-(morpholin-4-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}piperidin-2-one
1-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-3-(5-pentyl-1,3,4-thiadiazol-2-yl)urea
6-amino-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]pyridine-2-carboxamide
[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]methanamine
3-acetamido-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}benzamide
1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
2-[2-(3-fluorophenyl)ethyl]-4-[3-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 3-benzyl-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidine-3-carboxylate
N'1-(pentan-3-yl)-N'1-(2-phenylethyl)cyclopropane-1,1-dicarboxamide
ethyl 3-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propanoate
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-(oxan-2-ylmethyl)acetamide
N,1,7-trimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-indole-2-carboxamide