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3-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]-1-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)urea
3-methyl-4-[3-methyl-5-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
(2R,6S)-4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
5-(pentan-2-yl)-4-phenyl-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
3-ethoxy-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(2-chlorophenyl)methyl]-4-cyclobutanecarbonylmorpholine
{3-benzyl-1-[1-(3-chlorophenyl)piperidin-4-yl]piperidin-3-yl}methanol
3-(diphenylmethyl)-5-(2-methoxyethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-(2,3-dihydro-1H-indol-1-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
2-{2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
4-(4-methylphenyl)-3-[1-(pyrrolidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-N,N-bis(pyridin-4-ylmethyl)but-2-enamide
3-methyl-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)pyridin-2-amine
5-(methoxymethyl)-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
1-methyl-3-(2-methylpropyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
4-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyrimidine-5-carboxylic acid
4-(4-methoxyphenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazole
(1S,4S)-5-(2-amino-2-methylpropanoyl)-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-methyl-4-{2-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-2-yl]ethyl}piperazine
N-(2-chlorophenyl)-3-{[4-(3-hydroxypropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
N-(1-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)-2-(dimethylamino)-N-methylacetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(pyridin-3-yl)acetamide
2-methoxy-6-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
(1S,6R)-3-(2-oxo-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
6-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyrimidin-4-amine
1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-[2-(dimethylamino)ethyl]-N-ethyl-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
2,5-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-[4-(methylsulfanyl)phenyl]acetic acid
1-(dimethyl-1,3-thiazole-5-carbonyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-methyl-2-(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-3-oxopiperazin-2-yl)acetamide
(3S,4R)-4-(4-fluorophenyl)-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]pyrrolidine-3-carboxylic acid
7-methyl-2-[2-(thiophen-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-[1-(3-fluoropyridine-4-carbonyl)piperidin-4-yl]piperidin-4-ol
1-[4-(2-cyclopropyl-1H-imidazol-1-yl)butyl]azepane
7-[(2,4-dimethoxy-3-methylphenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}azetidin-3-yl)piperidine
(3S,4S)-4-methyl-1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-3,4-diol
N-cyclopentyl-2-methyl-N-(3-phenylprop-2-yn-1-yl)pyridine-3-carboxamide
3-(5-methylfuran-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
2-phenyl-4-[(3,4,5-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[5-({[(2-methoxyphenyl)methyl]carbamoyl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-(2H-1,3-benzodioxol-5-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]urea
N-{[2-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxy-2-methylpropan-1-one
4-fluoro-2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide