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(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-8-azabicyclo[3.2.1]octane
4-(cyclopropylmethyl)-1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-6-methylpyridazine
4-[benzyl({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]butan-1-ol
4-(3-hydroxy-3-methylbutyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
5-ethyl-N4-{2-[(2S)-pyrrolidin-2-yl]ethyl}pyrimidine-2,4-diamine
7-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(1R,5S,6S)-6-{[4-(2-chlorophenoxy)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
1-(4-ethoxyphenyl)-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
(3S,4S)-1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]pyridin-2-yl}-4-methylpiperidine-3,4-diol
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-2-(4-methanesulfonylphenyl)ethan-1-one
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4-(pyridin-4-yl)pyrimidin-2-amine
(2S,4R)-4-(dimethylamino)-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidine-2-carboxylic acid
1-amino-N-{[4-(methylsulfanyl)phenyl]methyl}-N-(prop-2-en-1-yl)cyclopropane-1-carboxamide
(1R,9aR)-1-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-cyclohexyl-2-oxo-2-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}acetamide
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-2,1,3-benzoxadiazole-4-sulfonamide
(3S,4S)-1-(2-amino-5-butyl-6-methylpyrimidin-4-yl)-4-[(dimethylamino)methyl]piperidin-3-ol
1-(pyrazine-2-carbonyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
methyl (2S,4R)-1-benzyl-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
4-methoxy-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-2-amine
4-{3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanoyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3,4-dihydropteridin-4-one
2-(2-fluoro-5-methoxyphenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
8-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-2-phenoxy-N-(pyrazin-2-ylmethyl)benzamide
1-{3-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]phenyl}ethan-1-one
N-benzyl-6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-sulfonamide
2-methyl-6-(1H-pyrazol-3-yl)quinoline
1-[1-(4-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)ethyl]pyrrolidine
2-(2,4-difluorophenyl)-5-(4,4,4-trifluorobutyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
4-cyclopentanecarbonyl-2-[(4-fluorophenyl)methyl]morpholine
1-[1-ethyl-5-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
4-[({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)methyl]-1,3-thiazol-2-amine
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
2-(3-fluoro-2-hydroxyphenyl)-1H-1,3-benzodiazole-6-carboxylic acid
N-[(1S)-1-phenylethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-(1-{7-[(4-acetamidophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-(3-methylbutyl)piperazin-2-yl)ethan-1-ol
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-3,5-dimethyl-1H-indole-2-carboxamide
N-[(1-propyl-1H-pyrazol-4-yl)methyl]-3-(pyrrolidine-1-sulfonyl)benzamide
6-oxo-1-propyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)piperidine-3-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2,5-dimethylfuran-3-carboxamide
7-(cyclopropylmethyl)-N-ethyl-6-(2-fluoro-4-methoxyphenyl)-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-5-methoxyphenol
2-{2-[6-methyl-5-(morpholine-4-carbonyl)-2-oxo-1,2,3,4-tetrahydropyrimidin-4-yl]phenoxy}acetic acid
(1S,5R)-3-(1H-1,3-benzodiazol-2-ylmethyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3aR,6aS)-5-[2-(morpholin-4-yl)benzoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-hydroxybenzamide
N-[3-(4-tert-butylphenoxy)-2-hydroxypropyl]-1,5-dimethyl-1H-pyrazole-4-carboxamide