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4-(4-hydroxy-4-phenylpiperidine-1-carbonyl)-1-(2-methylpropyl)pyrrolidin-2-one
N,N-dimethyl-5-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-cyclopentyl-N-propyl-3-(1H-pyrazol-4-yl)benzamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[(3S,4R)-3-methanesulfonamido-4-propylpyrrolidin-1-yl]acetamide
methyl 4-{[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)carbamoyl}butanoate
2-(1-benzofuran-5-yl)-1-(2-methanesulfonylethyl)-1H-imidazole
ethyl 2-{1-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]piperidin-2-yl}acetate
6-ethyl-2-(3-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-{4-phenyl-1-[3-(pyridin-3-yl)propyl]-1H-imidazol-5-yl}pyridine
1-{[(3R,4R)-4-(hydroxymethyl)-1-(6-methyl-2-propylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}piperidin-4-ol
1-(cyclohexylmethyl)-3-({[(2-fluorophenyl)methyl]amino}methyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
2-[4-(6-methylpyridazin-3-yl)-1H-pyrazol-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
3-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}-6-methyl-4H-chromen-4-one
1-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-ylmethyl]-1H-pyrazole-3-carboxylate
N-{2-[4-(dimethylamino)phenyl]ethyl}-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
4-{[1-cyclohexyl-5-(2-methanesulfonylethyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidine-2-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-[(dimethylamino)methyl]-1,3-thiazole-4-carboxamide
(2R,6R)-4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(4aR,8aS)-1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-decahydro-1,6-naphthyridin-6-yl]-2-(4-methoxyphenyl)ethan-1-one
N,N-dimethyl-3-({[(3-phenoxyphenyl)methyl]amino}methyl)pyridin-2-amine
N'-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-N,N-dimethylbutanediamide
1-[4-(4-fluorophenoxy)piperidine-1-carbonyl]-6-azaspiro[2.5]octane
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(1H-imidazol-4-yl)ethyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
2-(3-phenylpropyl)-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-5-carboxamide
1-(4-chloro-2-fluorophenyl)-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
1-methyl-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-1-{3-[(4-methylphenyl)sulfanyl]propyl}urea
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
2-benzyl-9-(propane-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
N3-[3-(4-hydroxyphenyl)propyl]piperidine-1,3-dicarboxamide
3-methyl-5-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazol-5-yl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-[2-(4-fluorophenyl)ethyl]-2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carboxamide
5-[1-(1-benzothiophene-2-carbonyl)piperidin-2-yl]-1-methyl-1,2,3,6-tetrahydropyridine
4-{[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
4-methyl-3-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]-2-propyl-2,5-dihydro-1H-pyrrole
2-[(2-fluorophenyl)methyl]-1,6-dimethyl-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N,2-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(thiophen-2-ylformamido)propanamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
(4aS,7aR)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
4-(2,3-dimethyl-1H-indole-7-carbonyl)-1-(3,5-dimethylphenyl)piperazin-2-one
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
ethyl 1-(2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}acetyl)piperidine-2-carboxylate
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(2,4-difluorophenyl)ethan-1-one
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-(1,2-oxazol-3-ylmethyl)-2-phenylacetamide
3-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)urea