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2-[4-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)morpholin-2-yl]ethan-1-ol
methyl 5-({4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}sulfonyl)-1-methyl-1H-pyrrole-2-carboxylate
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-phenylethane-1,2-dione
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(4-phenyl-1,3-thiazol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-1,3-benzodiazol-2-yl)ethan-1-ol
N-cyclopropyl-1-{1-[4-(4-hydroxyphenyl)butan-2-yl]piperidin-4-yl}piperidine-4-carboxamide
N-[3-(3-cyclohexyl-1,2,4-oxadiazol-5-yl)propyl]acetamide
1-methyl-4-(3-phenylpropyl)-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(2-methoxyphenyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
(4aS,8aR)-6-[(3-chloro-5-fluorophenyl)methyl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-N-(oxan-4-ylmethyl)-5-(phenoxymethyl)-1,2-oxazole-3-carboxamide
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3-(3-methylphenyl)piperidine
(1S,4S)-2-(4-chloro-2-methoxy-5-methylphenyl)-5-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-{1-[2-(dimethylamino)acetyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
N-[(2-fluorophenyl)methyl]-N-propylpiperidin-4-amine
3-acetamido-5-({[(3-fluorophenyl)methyl]amino}methyl)-N-(2-methoxyphenyl)benzamide
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,6-dimethylquinoline
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-methyl-N-[3-(piperidin-1-yl)propyl]propanamide
(2S,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N-{3-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]phenyl}methanesulfonamide
N-[4-(difluoromethoxy)phenyl]-3-(3-ethylphenoxy)azetidine-1-carboxamide
ethyl 2-{1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazol-3-yl]-N-methylformamido}acetate
(3aR,7aS)-N-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
6-cyano-N-[(3R,5S)-1-(2-ethoxyacetyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
2-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amine
3-{1-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1H-imidazol-2-yl}benzonitrile
(3-{2-[1-(2,3-dimethylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-[(3-{[2-(1H-imidazol-1-yl)ethyl]sulfamoyl}phenyl)formamido]-N,N-dimethylacetamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}piperidine
2-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
6-{1-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
N-cyclohexyl-1-cyclopropyl-5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
ethyl 3-(2-phenoxyethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxylate
N-[2-(diethylamino)ethyl]-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-6-methoxyphenol
{2-[(4aS,7aR)-4-benzyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}urea
N-(1H-1,2,4-triazol-5-ylmethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
1-(1-methylpiperidin-4-yl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-methyl-4-phenylpyrimidine-5-carboxamide
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]pyridine-3-carboxamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(6-hydroxy-6-methylheptan-2-yl)-1H-pyrazole-4-carboxamide
1-{3-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[benzyl(methyl)amino]-N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
6-{[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]methyl}-1,4-oxazepan-6-ol
4-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-N-phenylbenzamide
1-[(2,3-dimethoxyphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine