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N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
1-{[4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-4-ol
3-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
4,5-dimethyl 1-[(3S,5S)-5-[(1,3-dihydro-2-benzofuran-5-yl)carbamoyl]-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
3-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1-ethylpiperidine
2-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
3-(1-ethyl-1H-imidazol-2-yl)-1-[(4-methoxypiperidin-1-yl)sulfonyl]piperidine
3-[3-(4-chlorophenyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiolane-1,1-dione
1-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-methoxy-2-phenylethan-1-one
5-{[3-cyclopropyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-dimethylimidazolidine-2,4-dione
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
4,6-dimethyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-{3-[2-(2,5-dioxoimidazolidin-4-yl)acetamido]phenyl}-2-methoxybenzamide
2-[3-(2-methoxybenzoyl)piperidin-1-yl]pyridine-3-carboxamide
4-({3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
4-(2-fluorophenoxy)-1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]piperidine
N-cyclopropyl-1-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
6-ethyl-N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
7-chloro-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}quinolin-4-amine
1-[(5-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]azepane
1-[2-(3,5-dimethoxyphenyl)acetyl]-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
5-({[(3-{2-[4-(3,4-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
8-fluoro-2-[2-(3-methoxyphenyl)azetidine-1-carbonyl]quinoline
4-[(2-methoxyphenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
3-acetamido-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)benzamide
6-[2-(pyridin-2-ylsulfanyl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-ethyl-6-{4-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]piperazin-1-yl}pyrimidine
6-tert-butyl-1-methyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-methyl-N-{1-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
7-(cyclobutylmethyl)-2-(2-ethoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N,N-diethyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
2-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-N,N-bis(propan-2-yl)benzamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
2-[1-(2-methylphenyl)-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(1R,5R)-3-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-9-methyl-9H-carbazole-3-carboxamide
N,N-diethyl-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-amine
N-(3,3-diphenylpropyl)-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidine
2-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-1,3-benzoxazole
1'-[(4-methoxypyridin-2-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-ethyl-N-[2-(4-ethylmorpholin-2-yl)ethyl]-1H-pyrazole-4-sulfonamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-amine
2-(2,5-dimethylphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3ar,6ar)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-(1-methyl-1H-pyrrol-2-yl)-2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]ethane-1,2-dione
4-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[(2-methylpropyl)amino]methyl}piperidin-2-one