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1-(4-acetylphenyl)-3-{[1-(propan-2-yl)piperidin-3-yl]methyl}urea
2-(4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-(thiophen-2-yl)ethane-1,2-dione
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(furan-2-yl)propan-1-one
3-[2-(N-methylmethanesulfonamido)ethyl]-1-[2-(trifluoromethoxy)phenyl]urea
1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazole-4-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]-3-phenylpropan-2-ol
6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-2-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}urea
(2S,4R)-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-N-(diphenylmethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
3-(1H-pyrazol-1-ylmethyl)-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
3-[(4-fluorophenyl)formamido]-N-[(1-hydroxycyclohexyl)methyl]propanamide
N-{2-[(1-benzylpiperidin-4-yl)amino]ethyl}-N-methylmethanesulfonamide
4-[1-({[(2-methoxyphenyl)methyl]carbamoyl}methyl)piperidin-3-yl]benzoic acid
2,3-dimethyl-7-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane-6-carbonyl}-1H-indole
2-[4-(3-chlorothiophene-2-carbonyl)morpholin-3-yl]acetic acid
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
3-(isoquinolin-5-yl)-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}urea
1-{3-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-oxopropyl}piperidin-2-one
1-methyl-3-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-1-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
(4aS,8aR)-1-(2-aminoethyl)-6-[(4-methoxyphenyl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N,3,6-trimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
3-(5-{1-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
3-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)pyridine
3-(2,3-dichlorophenyl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
3-benzyl-1-(3-methoxypropyl)-8-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-[2-(6-methylpyridin-2-yl)ethyl]piperidin-4-amine
5-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
5-[1-(difluoromethyl)-1H-pyrazol-3-yl]-3-(thiophen-2-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
[(3-chlorophenyl)methyl]({[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
2-[(6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazin-3-yl)amino]ethan-1-ol
5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-2,1,3-benzothiadiazole
3-cyclopropyl-5-(5-fluoro-2-methoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
3-[(3R)-pyrrolidin-3-yl]-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
N-cyclopentyl-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-cyclohexyl-4-{3-[(3-methylpiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}piperazine
3-[(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridin-2-amine
2-(3-methoxypropyl)-9-(1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-(2-chloro-3-methylbenzoyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-methyl-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-pyrazole-5-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
methyl[(2-phenyl-1,3-thiazol-4-yl)methyl](3,3,3-trifluoropropyl)amine
N-[1-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
methyl (3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carboxylate
N-(4-{2-oxo-2-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethoxy}phenyl)propanamide
4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methylpyrimidin-2-amine
4-benzyl-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-6-[(5-methylthiophen-2-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-phenyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide