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1-(1H-imidazol-4-ylmethyl)-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
1-cyclopentyl-N3-methyl-N5-[(2-methylphenyl)methyl]-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-amino-1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-(1-phenoxypropan-2-yl)-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-cyclobutanecarbonyl-N-methyl-N-[3-(2-methylphenoxy)propyl]piperidine-4-carboxamide
3-(3-chlorophenyl)-1-[4-(hydroxymethyl)piperidin-1-yl]-3-(2-hydroxyphenyl)propan-1-one
2-(5-methyl-1,2-oxazol-3-yl)-N-(2-methyl-5-sulfamoylphenyl)piperidine-1-carboxamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-methanesulfonylpiperidin-4-amine
N-[2-(N-methylmethanesulfonamido)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidine-3-carboxylic acid
(1H-imidazol-2-ylmethyl)[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amine
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
2-methyl-3-[5-(2-methylpyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]propanoic acid
N-methyl-N-[2-(morpholin-4-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
2-[(3,4-dimethoxyphenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-methylphenyl)piperidine
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-(oxan-4-yl)piperidine
2,6-dimethyl-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
14-(2-chloro-3,4-dimethoxyphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-acetyl-N-(4-chloro-2-ethylphenyl)-1,4-diazepane-1-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
1-methyl-4-[2-(pyrazin-2-yloxy)hex-5-en-1-yl]-1,4-diazepane
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-{4-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]benzamide
2-(3-methoxypropyl)-8-[3-(pyridin-3-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
7-[2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
3-{[(2-carbamoylethyl)(propan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
2-methoxy-3-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}pyridine
(4aR,8aS)-1-(2,6-difluorobenzoyl)-N,N-dimethyl-decahydro-1,6-naphthyridine-6-sulfonamide
N-[3-({[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}methyl)-5-(piperidine-1-carbonyl)phenyl]methanesulfonamide
N-[cyclopropyl(4-methoxyphenyl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
9-[(2S)-2-amino-4-(methylsulfanyl)butanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-2-[4-(9H-purin-6-yl)-1H-pyrazol-1-yl]acetamide
2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
[(3R,4R)-1-(5-ethyl-1H-pyrrole-2-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
6,8-dimethoxy-4-methyl-2-[3-(3-methylphenoxy)azetidin-1-yl]quinoline
N-(3-cyano-4-methylphenyl)-3-(propoxymethyl)pyrrolidine-1-carboxamide
(1R,3S,5S)-8-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-3-(3-methylfuran-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-ethyl-3-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
2-(dimethylamino)-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-2-(3-methylphenyl)acetamide