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2-[4-(3-chloropyridin-2-yl)-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(4-fluorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
N-[1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidin-3-yl]acetamide
2-(4-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenoxy)ethan-1-ol
7-(3-fluoro-4-methoxyphenyl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
methyl 3-(1-phenylcyclopropaneamido)-6-(piperidin-1-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
4-(2,5-dimethoxyphenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenol
5-chloro-3-[2-(3-methoxypropyl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
(2R)-2-[5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
1-(4,4,4-trifluorobutyl)-1,2-dihydroquinolin-2-one
2-[1-methyl-4-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperazin-2-yl]ethan-1-ol
7-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-[3-(pyridin-2-yl)propyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl}){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
1-{1-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
5-methyl-1-[2-oxo-2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-phenyl-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-pyrazole-4-carboxamide
methyl 2-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-3-carboxylate
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
(2E)-3-(3,4-dimethoxyphenyl)-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)prop-2-enamide
N-[(3R,4R)-3-hydroxy-1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl]pyrazine-2-carboxamide
1-(2,3-dimethoxybenzoyl)-3-(2-methoxybenzoyl)piperidine
2-(4-methylphenyl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
2-ethyl-8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-4-(pyridin-2-yl)pyrimidine
2-benzyl-9-[2-(propylsulfanyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3S,5R)-1-[2-chloro-5-(trifluoromethyl)benzoyl]-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
1-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]pyrrolidin-2-one
N-[(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
5-[2-(2-{[4-(ethylamino)pyrimidin-2-yl]amino}ethyl)morpholin-4-yl]-2-methyl-2,3-dihydropyridazin-3-one
4-(1H-imidazol-1-yl)-1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}butan-1-one
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
6-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyridine-3-carbonitrile
2-(2-chlorophenyl)-1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
3-(3-fluorophenyl)-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperazin-2-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,N,5-trimethylthieno[2,3-d]pyrimidine-6-carboxamide
1'-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
5-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
4-(1H-indol-3-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]butan-1-one
1-(but-3-enoyl)-N-[3-(3-chlorophenyl)phenyl]piperidine-4-carboxamide
3-{[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
3-{[(3-methylthiophen-2-yl)methyl]amino}-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]benzamide
N-ethyl-3-{[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]sulfamoyl}-N-methylbenzamide
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyrazin-2-ol
1-methyl-8-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
N-[3-methyl-1-(4-methylphenyl)-1H-pyrazol-5-yl]-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide