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3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(oxolan-2-ylmethyl)-N-propylpropanamide
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-(6-methoxynaphthalene-2-carbonyl)piperidine
[1-(3-chloro-4-fluorobenzenesulfonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
2-(3-methyl-1,2-oxazol-5-yl)-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-acetamidoacetamide
N-(thiophen-2-ylmethyl)-6-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-(5-methylfuran-2-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-(3-phenylpropyl)piperidine-4-carboxylic acid
1-(2,6-dimethylpyridin-4-yl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazine
4-[2-(propylsulfanyl)pyrimidin-5-yl]-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-(4-methanesulfonylphenyl)-N-(propan-2-yl)pyrimidin-4-amine
2-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(isoquinolin-1-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
(2R,3R,6R)-5-(4-fluorobenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{2-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
methyl 2-{2-[2-(cyclopropylcarbamoyl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}acetate
(4aR,7aS)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[(2E)-2-ethylbut-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-[(dimethylcarbamoyl)methyl]-N-(3-fluorophenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[3-(dimethylamino)phenyl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide
(2S)-2-amino-N-(1-methylpiperidin-4-yl)-4-(methylsulfanyl)-N-(pyridin-4-ylmethyl)butanamide
(2S)-N-cyclopropyl-2-(methylamino)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
dimethyl(2-{2-[3-(piperidine-1-carbonyl)phenyl]phenoxy}ethyl)amine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-2-ol
1,3,6-trimethyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-fluoro-4-hydroxybenzamide
1-methyl-5-(1-methyl-4-phenyl-1H-imidazol-5-yl)-1H-indole
N,N-dimethyl-5-[methyl(2-phenylethyl)amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]methyl}furan-2-carboxamide
ethyl(oxan-4-ylmethyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-(1-cycloheptylpiperidin-3-yl)-2-methoxybenzene-1-sulfonamide
4-[4-(3-aminopentan-3-yl)-1H-1,2,3-triazol-1-yl]-N-cycloheptylpiperidine-1-carboxamide
1-[7-(5-fluoropyrimidin-2-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-4-ol
methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
1-(3-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}phenyl)ethan-1-one
(3R,4S)-4-(5-methylfuran-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-3-amine
2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
2-[(2-fluorophenyl)methyl]-1,6-dimethyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
methyl[(1-{[1-(oxane-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
4-[(2S)-1-acetylpyrrolidine-2-carbonyl]-1-(4-methylphenyl)piperazin-2-one
2-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
ethyl 1-(4-hydroxy-4-methylpentan-2-yl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
1-[2-(dimethylamino)ethyl]-4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one