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3-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
(2S)-2,6-diamino-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]hexan-1-one
3-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl]benzonitrile
4-[(6-methylpyridin-3-yl)oxy]-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
5-(2-cyclopropylpyrimidin-4-yl)-2-ethoxybenzoic acid
4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
2-(3-{[(2R,3S,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenoxy)ethan-1-ol
N'-benzyl-N-cyclopentyl-N'-(2-hydroxyethyl)butanediamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
3-{[(2R)-2-methylpiperazin-1-yl]sulfonyl}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
4-[(2-methylphenyl)methyl]-1-(2-methylpropyl)-1,4-diazepan-5-one
5-methoxy-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyrimidine
N-cyclopropyl-3-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}propanamide
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]urea
1-{2-[(2-methylprop-2-en-1-yl)oxy]benzamido}piperidine-3-carboxylic acid
3-{[1-(1-phenylcyclopentanecarbonyl)pyrrolidin-3-yl]methyl}benzamide
3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
3-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-1-(propan-2-yl)piperidine-4-carboxamide
(2R)-2-hydroxy-1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-2-phenylethan-1-one
(3R,4S)-4-cyclopropyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-amine
2-{1-[1-(thiophene-3-sulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
9-[(3-fluoro-4-methoxyphenyl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-({[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)pyrimidin-4-ol
N-methyl-2-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}amino)pyridine-4-carboxamide
N,5-dimethyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
(3aS,6aS)-2-(1H-imidazol-4-ylmethyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-1-(2-phenylphenyl)piperazin-2-one
4'-[2-(4-fluorophenoxy)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1S,6R)-3-({3-[4-(morpholin-4-yl)butoxy]phenyl}methyl)-3,9-diazabicyclo[4.2.1]nonane
N-[(4-fluorophenyl)methyl]-1-methyl-5-[(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S)-1-(6-methoxypyridine-3-carbonyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-fluorophenyl)ethyl]piperidine
2-(azepan-1-yl)-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
methyl({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(oxan-2-ylmethyl)amine
4-{5-[1-(difluoromethyl)-1H-pyrazol-3-yl]-3-methyl-1H-1,2,4-triazol-1-yl}-2-methylpyridine
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-(4-{[(2-phenoxypyridin-3-yl)methyl]amino}piperidin-1-yl)ethan-1-one
N-(1,3-benzothiazol-2-ylmethyl)-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-methyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-5-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-N-(pentan-3-yl)-N-(2-phenylethyl)propanamide
2-ethyl-N-[2-(4-fluorophenyl)ethyl]-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propanoic acid
N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1,9-dioxaspiro[5.5]undecan-4-amine
(4aR,7aS)-1-benzyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)oxolane-2-carboxamide
3-(4-methylpiperazine-1-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine