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5-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
6-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-4-oxo-4H-pyran-2-carboxamide
1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-[2-(dimethylamino)-2-(4-fluorophenyl)ethyl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
N-[(4-methoxypyridin-2-yl)methyl]-4-methyl-1H-imidazole-2-carboxamide
methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
[(2,4-difluoro-3-methoxyphenyl)methyl](propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-(1H-1,3-benzodiazol-1-yl)-1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}ethan-1-one
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
5-(2-{1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)-4,6-dimethylpyrimidin-2-ol
2-[2-(1H-imidazol-4-yl)ethyl]-9-(pyrrolidine-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
8-({5-methanesulfonyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-cyclopropylacetyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
3,5-dimethyl-4-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
N-ethyl-2,2,3,3-tetramethyl-N-[2-(pyrrolidin-1-yl)ethyl]cyclopropane-1-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2,5-dimethoxyphenyl)-3-(oxan-4-yl)-4H-1,2,4-triazole
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-2-(1H-imidazol-2-yl)benzamide
1-(3,5-dimethylphenyl)-4-(1-methyl-2-oxoimidazolidine-4-carbonyl)piperazin-2-one
methyl({[6-(3-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})(1H-pyrazol-3-ylmethyl)amine
1-[(1S,5R)-6-[6-(dimethylamino)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
14-(1H-indol-2-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
5-{methyl[(3-methylpyridin-4-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-oxoacetamide
(2S,4S)-N-ethyl-1-(1-methylpiperidin-4-yl)-4-[2-(pyridin-4-yl)acetamido]pyrrolidine-2-carboxamide
N-{3-[5-(piperazin-1-ylmethyl)thiophen-3-yl]phenyl}acetamide
5-cyclobutanecarbonyl-1'-(3-fluoropyridin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)methanol
4-ethyl-5-methyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}pyrimidin-2-amine
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-(4-methylphenyl)pyridine-3-carbonitrile
N-(furan-2-ylmethyl)-1-(2-methylpropyl)-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}azepane
6-methyl-5-[5-({[2-(pyrrolidin-1-yl)ethyl]sulfanyl}methyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-{1-[2-(1,2-benzoxazol-3-yl)acetyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
(1R,5R)-3-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,9-diazabicyclo[3.3.2]decan-10-one
1-(3-methoxyphenyl)-4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazin-2-one
2-{4-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
4-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1,3-oxazole-5-carboxamide
7-fluoro-1-[(3-methoxyphenyl)methyl]-3-({methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(3-cyclopentylpropyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
4-{2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-(1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)ethan-1-ol
N-[(2-chloro-6-fluorophenyl)methyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-[3-(4-methylphenyl)propyl]-2-(1-methylpiperidin-2-yl)acetamide
3-benzyl-8-[(4-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-{3-[4-(piperidine-1-carbonyl)phenyl]phenyl}-1H-pyrazol-1-yl)acetamide
2-(dimethyl-1,3-thiazol-4-yl)-N-[(4-methoxyphenyl)methyl]-N-propylacetamide
N-(butan-2-yl)-2,3-dimethoxy-N-(pyridin-4-ylmethyl)benzamide