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1-({[(3-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}-4-methoxyphenyl)methyl]amino}methyl)cyclohexan-1-ol
N-benzyl-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
8-chloro-2-[1-(2-methanesulfonylethyl)-1H-1,2,3-triazol-4-yl]quinoline
3-(1H-1,3-benzodiazol-1-yl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-(thiophen-2-yl)-1H-imidazole
2-[5-cyclopropyl-4-(4-methylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(5-methylfuran-2-yl)pyrimidine
(3aS,6aS)-5-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-(5,6,7,8-tetrahydroquinoxalin-5-yl)benzamide
1-[4-({[(1-benzyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)thiophen-2-yl]ethan-1-one
6-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-2-(2-methoxyethyl)piperidine
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-methyl-1-benzofuran-2-carboxamide
2-(1-phenylethyl)-1-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-imidazole
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-cyclopropylacetamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(5-fluoro-1H-1,3-benzodiazol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(2-methoxyphenyl)methyl]-5-methyl-6-[2-(pyridin-3-yl)piperidine-1-carbonyl]thieno[2,3-d]pyrimidin-4-amine
[(3R,4R)-1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
1-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(oxolan-2-ylmethyl)piperazine
methyl 3-cyclobutaneamido-5-[(cyclohex-3-en-1-ylmethyl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl][(5-ethylpyridin-2-yl)methyl]methylamine
N-(2-methoxyethyl)-N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
3-(3-methoxypropyl)-1-[(3-methylpyrazin-2-yl)methyl]piperidine-3-carboxylic acid
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3R,4R)-1-(3-cyano-2-methoxypyridin-4-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
5-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(4-cyclopentylphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-(4-methoxyphenyl)-1,2,4-triazin-3-amine
N-ethyl-6-(3-fluorophenyl)-N-(2-methylprop-2-en-1-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[2-(4-sulfamoylphenyl)ethyl]-3-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
(2R,3R)-3-(2-methyl-1H-imidazol-1-yl)-1'-(thiophen-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1-methyl-1H-imidazol-2-yl)({1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl})methanol
1-[cyclohexyl(methyl)amino]-3-(4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-cyclopentyl-1-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-2-phenylethan-1-one
4-[(diethylamino)methyl]-5-ethyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]furan-2-carboxamide
2-methyl-3-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine-1-carbonyl}pyridine
N-(3-cyclopentylpropyl)-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-benzoyl-1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)piperidine
1-methyl-3-(1-methyl-3-phenyl-1H-1,2,4-triazol-5-yl)piperidine
2-methyl-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)[3-(1H-pyrazol-1-yl)propyl]amine
N-[3-(4-hydroxyphenyl)propyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-1H-imidazol-2-yl}-1-methyl-1H-1,3-benzodiazole
(1S,5R)-3-[2-(3-chloro-4-fluorophenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-ethyl-4-[(1-methylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
4-[5-(2-aminoethyl)-2-methoxyphenyl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(2S,4R)-N,N-diethyl-1-(3-methylbut-2-en-1-yl)-4-(5-methylthiophene-2-amido)pyrrolidine-2-carboxamide