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5-methyl-N-[(6-methylpyridin-2-yl)methyl]-6-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}thieno[2,3-d]pyrimidin-4-amine
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(oxan-2-ylmethyl)-1,3-oxazole-4-carboxamide
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 4-methyl-3-({3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}amino)benzoate
1-(2-methoxyethyl)-3,8-bis(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(thiophen-3-ylmethyl)propanamide
(1S,5R)-6-propyl-3-(2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-(1,2-oxazol-3-ylmethyl)benzamide
5-(pyridin-2-yl)-5-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[1-(5-cyanopyridin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-phenylpyrimidin-4-ol
3-{2-oxo-2-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}imidazolidine-2,4-dione
3-(methylsulfanyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-({4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
2-(2-methoxyethyl)-8-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(1H-imidazol-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
3-(1-butyl-1H-imidazol-2-yl)-1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
2-(4-{[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
N,N-bis(prop-2-en-1-yl)-3-(quinolin-5-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-cyano-N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)benzamide
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
({5-[4-(ethanesulfonyl)piperazine-1-carbonyl]-1,3,4-oxadiazol-2-yl}methyl)dimethylamine
8-chloro-2-({[(1-ethyl-1H-indazol-3-yl)methyl]amino}methyl)quinolin-4-ol
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-methyl-2-(3-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
1-[(3-ethoxy-2-hydroxyphenyl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
N-(1,4-dioxan-2-ylmethyl)-5-(2-methylphenyl)-1,2,4-triazin-3-amine
(3S,4S)-1-(5-methylthiophene-2-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}({[2-(1H-pyrazol-1-yl)phenyl]methyl})amine
3-benzyl-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
5-{1-[1-(furan-2-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}-2-methoxyphenol
3-(1H-imidazol-1-ylmethyl)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
N-{[(2S,4S)-4-fluoro-1-(3-hydroxypyridine-2-carbonyl)pyrrolidin-2-yl]methyl}pyridine-3-sulfonamide
2-(cyclopropylamino)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-1,3-dimethyl-N-[(3S)-2-oxoazepan-3-yl]-1H-pyrazole-5-carboxamide
1-[2-methoxy-4-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
4-(5-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazol-2-yl)morpholine
(2S,4S)-1-(2,2-diphenylethyl)-N-methyl-4-{[(2,3,4-trimethoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-methyl-N-[1-(1-{spiro[2.4]heptane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-(cyclopropylmethyl)-3-(6-methoxynaphthalene-2-carbonyl)piperidine
2-cyclobutyl-1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
8-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(4-cyano-2-ethylphenyl)-3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]urea
5-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyrazin-2-ol
N-[(5-methylfuran-2-yl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
6-(3-fluorophenyl)-N-methyl-N-(oxan-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N,N-dimethyl-6-({1-[methyl(pyridin-3-ylmethyl)amino]hex-5-en-2-yl}oxy)pyrazin-2-amine