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(8R,9aS)-8-hydroxy-2-[3-(morpholin-4-yl)propyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
2-(2-{[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2,5-dihydro-1H-pyrrol-2-yl)methanol
2-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N,N-dimethylacetamide
(3S,4R)-3-methoxy-1-(1,8-naphthyridine-2-carbonyl)piperidin-4-amine
N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(1,3-thiazol-2-ylmethyl)acetamide
6-({[(4-phenyloxan-4-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4R)-1-(2-amino-1,3-benzothiazole-5-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-(oxane-2-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
4-fluoro-N-(2-{[1-(2-methoxyacetyl)piperidin-3-yl]formamido}ethyl)benzamide
1-[4-(2-fluoro-6-methoxyphenyl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,3,5-trimethyl-1H-indole-2-carboxamide
9-[(3,4-dimethylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4,5,6,7-tetrahydro-2H-indazole
(1S,3R)-3-amino-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)cyclopentane-1-carboxamide
N-[4-({[2-(piperidin-1-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
3-(2H-1,3-benzodioxol-5-yl)-1-[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]propan-1-one
(1S,5R)-3-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(3,5-difluorophenyl)methyl]-8-(piperidin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
5-{[benzyl(methyl)amino]methyl}-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)pyridine-4-carboxamide
N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]propanamide
methyl N-[1-oxo-1-(3-oxo-4-phenylpiperazin-1-yl)propan-2-yl]carbamate
2-amino-4-[(1H-indol-4-ylmethyl)amino]quinazoline-6-carboxylic acid
2-(3-benzoylpiperidine-1-carbonyl)-5-fluoro-1,3-dimethyl-1H-indole
{2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}urea
1-(1H-indazol-6-yl)-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1λ6-thiomorpholine-1,1-dione
(5S,9aS,9bS)-5-(2H-1,3-benzodioxol-4-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(benzylsulfamoyl)[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]amine
N-{4-[({[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}carbamoyl)methoxy]phenyl}propanamide
(1S,5R)-6-(cyclobutylmethyl)-3-(2-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]propanamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(thiophene-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{2,4,6-trimethyl-3-[({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}amino)methyl]phenyl}methyl acetate
1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(4-phenylphenyl)ethan-1-one
methyl(1,2-oxazol-3-ylmethyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-[5-(morpholin-4-ylmethyl)pyridin-2-yl]benzoic acid
(3S,4S)-1-[3-(piperidin-4-ylmethyl)benzoyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
N-methyl-2-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyridine-3-carboxamide
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-2-(pyridin-3-yl)acetamide
5-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-2-methoxyphenol
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N,N-dimethyl-1H-pyrazole-4-carboxamide
N-methyl-N-(propan-2-yl)-2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-[1'-(2,1,3-benzoxadiazol-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
6-ethyl-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrimidin-4-amine
4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1λ6-thiomorpholine-1,1-dione