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N-({4-hydroxy-1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]azepan-4-yl}methyl)pyrrolidine-1-carboxamide
1-[4-({[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}amino)piperidin-1-yl]ethan-1-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-cyclobutanecarbonyl-4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidine
methyl 2-(2-methoxy-4-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}phenoxy)acetate
2-methyl-3-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-N-(pyridin-3-ylmethyl)aniline
N-[(5-fluoro-2-methylphenyl)methyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(pyridin-2-ylmethyl)-4-[4-(trimethyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-cyclopentyl-N'-methyl-N'-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanediamide
N-ethyl-2-[(E)-2-phenylethenyl]pyrimidin-4-amine
N-[(2S)-1-hydroxypropan-2-yl]-6-(4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridin-3-ol
(2S,4S)-4-amino-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2,4-dimethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1,3-thiazole-5-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
2-(4-{[4-(benzyloxy)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
(1S,2S,9S)-N-(2-methoxy-6-methylphenyl)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]quinoxaline
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
1-(4-methylphenyl)-4-(3-phenylpropanoyl)piperazin-2-one
(2-methoxyethyl)(methyl)[(2-phenyl-1H-imidazol-4-yl)methyl]amine
1-{2-[4-(2-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
3-{1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
2-{4-[(ethylcarbamoyl)methyl]piperazin-1-yl}-6-phenylpyridine-3-carboxylic acid
2-(4-fluoro-3-methylphenyl)-2-[methyl(2-phenoxyethyl)amino]acetic acid
2-({4-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
3-(2-ethoxyphenyl)-6-(pyrrolidin-1-yl)pyridazine
1-(3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)-2-(2-methoxyethyl)piperidine
2-(2-hydroxyethyl)-8-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
methyl (1S,3R,3aR,6aS)-5-methyl-4,6-dioxo-1-phenyl-3-[2-(1H-pyrazol-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[6-(1-benzothiophen-7-yl)pyridin-2-yl]piperazine
N-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-N-methylthian-4-amine
5-(2-chloro-4-methoxyphenoxymethyl)-N-[3-(methylsulfanyl)propyl]-1,2-oxazole-3-carboxamide
4-(pyridin-3-yl)-6-(3,4,5-trifluorobenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-1,2,3-benzotriazole-5-carboxamide
1-(2,3-dimethylphenyl)-4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
N-cycloheptyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-cyclopropyl-1-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
(1R,3S)-3-methoxy-7-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
4-[(2R,5R)-2,5-dimethyl-4-(prop-2-en-1-yl)piperazin-1-yl]pyrimidine-5-carboxylic acid
3-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
1-[(3-methoxyphenyl)methyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
1-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
1-{4-[2-(morpholin-4-yl)ethyl]piperazin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
5-[1-(methoxymethyl)cyclobutanecarbonyl]-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(3,5-difluoro-4-methoxyphenyl)pyridine-3-carbonitrile
2-[ethyl(pyridin-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
8-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid