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7-cyclopropanecarbonyl-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperidin-4-yl]piperidin-4-ol
1-[3-({2-[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]-1H-imidazol-1-yl}methyl)piperidin-1-yl]ethan-1-one
3-{[1-butyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3,3-dimethylurea
2-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-[methyl(1,2-oxazol-3-ylmethyl)amino]-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
methyl 3-[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)carbamoyl]propanoate
5-{[4-(2,6-dimethoxypyrimidin-4-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
1-{4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-[5-(3-chloro-4-fluorobenzoyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-[4-(2-fluorophenoxy)phenyl]-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
N,N-dimethyl-5-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}-1,3-thiazol-2-amine
4-(4-fluorophenyl)-5-methyl-2-(4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-(propan-2-yl)-1H-pyrazol-1-yl)pyrimidine
2-tert-butyl-7,7-dimethyl-N-(propan-2-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
4-(2-ethoxypyridine-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
N-(2-chloropyridin-3-yl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
4-[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridine-2-carbonyl]benzonitrile
N6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-9H-purine-2,6-diamine
ethyl 1-{[(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-imidazole-2-carboxylate
8-[4-(trifluoromethyl)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
1-methyl-6-(propan-2-yl)-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-dihydropyridin-2-one
methyl({[5-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
3-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-1-(2-methoxyphenyl)urea
{[7-chloro-2-(2-phenylethoxy)quinolin-3-yl]methyl}[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-methyl-3-(1H-pyrazol-1-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
1-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-(5-ethoxyfuran-2-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
4-[(1S,2R)-2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1-hydroxypropyl]phenol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]amine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
8-(oxan-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
[(2-chloro-6-fluorophenyl)methyl](methyl)[2-(pyridin-4-yl)ethyl]amine
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}thiophene-2-carboxamide
(3aS,6aS)-5-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N5-(3-methoxypropyl)-N6-{[1-(propan-2-yl)piperidin-3-yl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
5-(furan-2-yl)-3-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
2-{[methyl(quinolin-2-ylmethyl)amino]methyl}benzoic acid
2-methyl-5-{[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]sulfanyl}-1,3,4-thiadiazole
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methoxy-3-(morpholin-4-yl)benzamide
3-(pyridin-3-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-(4-methylphenyl)-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazin-2-one
1-{[methyl(1H-pyrazol-3-ylmethyl)carbamoyl]methyl}piperidine-4-carboxamide
1-(2-{[(2-hydroxyethyl)(methyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2-[3,5-dimethyl-4-(quinolin-6-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
1-(2-aminoethyl)-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-1H-1,2,3-triazole-4-carboxamide
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine
2-(methylsulfanyl)-1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)ethan-1-one
N-cyclopentyl-2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide